Browse Items (5 total)
- Tags: Competitive
Neurokinin-1 receptor resensitization precedes receptor recycling.
Tags: 2005, Adenosine Triphosphate/pharmacology, Animals, Bennett V J, Binding, Calcium/metabolism, CHO Cells, Competitive, Cricetinae, Guanylyl Imidodiphosphate/pharmacology, Neurokinin-1/*metabolism, Perrine S A, Phosphorylation, Rats, Receptors, Simmons M A, Substance P/metabolism, The Journal of pharmacology and experimental therapeutics
Multiple binding sites for [125I]RTI-121 and other cocaine analogs in rat frontal cerebral cortex.
Tags: *Membrane Transport Proteins, *Nerve Tissue Proteins, *Symporters, 1998, Animals, Binding, Binding Sites, Boja J W, Carrier Proteins/*metabolism, Carroll F I, Cocaine/*analogs & derivatives/pharmacokinetics, Competitive, Corpus Striatum/*metabolism, Dopamine Plasma Membrane Transport Proteins, Dopamine/metabolism, Frontal Lobe/*metabolism, Iodine Radioisotopes/*pharmacokinetics, Kinetics, Kopajtic T, Kuhar M J, Male, Membrane Glycoproteins/*metabolism, Norepinephrine Plasma Membrane Transport Proteins, Norepinephrine/metabolism, Rats, Regression Analysis, Serotonin Plasma Membrane Transport Proteins, Serotonin/metabolism, Sprague-Dawley, Synapse (New York, N.Y.), Vaughan R A
Virtual screening to identify novel antagonists for the G protein-coupled NK3 receptor.
Tags: *Models, *Narcotic Antagonists, *Quantitative Structure-Activity Relationship, 2010, Animals, Binding, Calcium Signaling/drug effects, CHO Cells, Competitive, Cricetinae, Cricetulus, Databases, Factual, Geldenhuys Werner J, Humans, Journal of medicinal chemistry, Kuzenko Stephanie R, Ligands, Molecular, Neurokinin-3/*antagonists & inhibitors/chemistry, Opioid/chemistry, Quinolines/*chemistry/pharmacology, Radioligand Assay, Receptors, Simmons Mark A
Binding of sequence-specific proteins to the 3'-untranslated region of vasoactive intestinal peptide mRNA.
Tags: 1995, Animals, Anterior/*metabolism, Base Sequence, Binding, Biochemical and biophysical research communications, Competitive, Cytoplasm/chemistry, Gene Expression Regulation, Genomic Library, Male, Messenger/*metabolism, Molecular Sequence Data, Pituitary Gland, Post-Transcriptional, Protein Binding, Proto-Oncogene Proteins c-fos/genetics, Rats, RNA, RNA Processing, RNA-Binding Proteins/*metabolism, RNA/metabolism, Signs S A, Sprague-Dawley, Subcellular Fractions, Tissue Distribution, Vasoactive Intestinal Peptide/*genetics, Wolford J K
Transcriptional regulation of human oxysterol 7 alpha-hydroxylase gene (CYP7B1) by Sp1.
Tags: 2001, Base Sequence, Binding, Binding Sites/genetics, Cell Line, Chiang J Y, Competitive, CpG Islands/genetics, Cultured, Cytochrome P-450 Enzyme System/*genetics/metabolism, Cytochrome P450 Family 7, Department of Integrative Medical Sciences, DNA/genetics, Enzymologic, gene, Gene Expression Regulation, Genetic, Humans, Luciferases/genetics/metabolism, Molecular Sequence Data, Mutagenesis, NEOMED College of Medicine, Nucleic Acid/genetics, Protein Binding, Recombinant Fusion Proteins/genetics/metabolism, Regulatory Sequences, Sequence Deletion, Site-Directed, Sp1 Transcription Factor/metabolism/*physiology, Steroid Hydroxylases/*genetics/metabolism, Transcription, Transfection, Tumor Cells, Wu Z