Browse Items (132 total)
- Tags: Dose-Response Relationship
The effect of GDNF on nigrostriatal dopaminergic function in response to a two-pulse K(+) stimulation.
Tags: *Nerve Growth Factors, 2000, 3, 4-Dihydroxyphenylacetic Acid/metabolism, Animals, Corpus Striatum/*drug effects/metabolism, Dluzen D E, Dopamine/*metabolism, Dose-Response Relationship, Drug, Experimental neurology, Extracellular Space/metabolism, Glial Cell Line-Derived Neurotrophic Factor, Male, Microdialysis, Nerve Tissue Proteins/*pharmacology, Neuroprotective Agents/*pharmacology, Parkinson Disease/drug therapy/metabolism, Potassium/*pharmacology, Rats, Sprague-Dawley, Substantia Nigra/*drug effects/metabolism, Xu K
Formulation and photoirradiation parameters that influenced photoresponsive drug delivery using alkoxylphenacyl-based polycarbonates.
Tags: 2014, Animals, Biocompatibility, Cardiotoxicity, Cell Line, Chamsaz Elaheh A, Chemistry, Department of Pharmaceutical Sciences, Dose-Response Relationship, Doxorubicin, Drug, Drug Delivery Systems/*methods, European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V, Heart/drug effects, Humans, Inbred BALB C, Joy Abraham, Mice, Nanotechnology, NEOMED College of Pharmacy, Oyewumi Moses O, Pharmaceutical, Photic Stimulation/*methods, Photoresponsive, Photosensitizing Agents/*chemical synthesis/radiation effects/toxicity, Polycarboxylate Cement/*chemical synthesis/radiation effects/toxicity, Polymer chain scission, Stimuli-responsive, Tumor, Wehrung Daniel
Antitumor efficacy and tolerability of systemically administered gallium acetylacetonate-loaded gelucire-stabilized nanoparticles.
Tags: *Lethal Dose 50, 2013, Adenocarcinoma/*drug therapy/pathology, Animals, Antineoplastic Agents/administration & dosage/pharmacokinetics/toxicity, Bi Lipeng, Cell Line, Department of Pharmaceutical Sciences, Dose-Response Relationship, Drug, Drug Stability, Drug Tolerance, Gallium/*administration & dosage/pharmacokinetics/*toxicity, Geldenhuys Werner J, Humans, Journal of biomedical nanotechnology, Metabolic Clearance Rate, Mice, Nanocapsules/*administration & dosage/chemistry/*toxicity, NEOMED College of Pharmacy, Nude, Organ Specificity, Oyewumi Moses O, Tissue Distribution, Treatment Outcome, Triglycerides/chemistry, Tumor, Wehrung Daniel
Efficacy of Higher-dose Oseltamivir in Adults with Influenza A and B.
Tags: 2014, Department of Internal Medicine, Dose-Response Relationship, Infectious Disease Alert, Influenza – Drug Therapy, Influenza A Virus, Influenza B Virus, Multicenter Studies, NEOMED College of Medicine, Oseltamivir – Adverse Effects, Oseltamivir – Therapeutic Use, Prospective Studies, Treatment Outcomes, Watkins Richard R
Steroids Increase the Risk for Community-acquired Staphylococcus aureus Bacteremia...Smit J, Kaasch AJ, Sogaard M , t al. Use of glucocorticoids and risk of community-acquired Staphylococcus aureus bacteremia:A population-based case-control study. Mayo Clin Proc 2016 :91:873-880.
Tags: 2016, Bacteremia – Risk Factors, Community-Acquired Infections – Risk Factors, Denmark, Department of Internal Medicine, Dose-Response Relationship, Drug, Glucocorticoids – Adverse Effects, Infectious Disease Alert, NEOMED College of Medicine, Staphylococcal Infections – Risk Factors, Staphylococcus aureus, Watkins Richard R
Antitumor activities of extracts from selected desert plants against HepG2 human hepatocellular carcinoma cells.
Tags: 2013, Aerial, Antineoplastic Agents, Bishayee Anupam, Carcinoma, Desert Climate, Dose-Response Relationship, Drug, Harlev Eli, Hep G2 Cells, Hepatocellular/*drug therapy/pathology, Humans, Inhibitory Concentration 50, Liver Neoplasms/*drug therapy/pathology, Mandal Animesh, Medicinal/chemistry, Nevo Eviatar, Pharmaceutical biology, Phytogenic/administration & dosage/*pharmacology, Plant Components, Plant Extracts/administration & dosage/*pharmacology, Plants, Tetrazolium Salts/chemistry, Thiazoles/chemistry, Thoppil Roslin J, Time Factors
Selective Targeting of Heme Protein in Cytochrome P450 and Nitric Oxide Synthase by Diphenyleneiodonium.
Tags: *cytochrome P450, *flavoenzymes, *heme, *nitric oxide synthase, *Reactive oxygen species, 2016, Aleksunes Lauren M, Animals, Cytochrome P-450 Enzyme Inhibitors/*pharmacology, Cytochrome P-450 Enzyme System/*metabolism, Department of Pharmaceutical Sciences, Dose-Response Relationship, Drug, Heck Diane E, Heindel Ned D, Heme/*antagonists & inhibitors/metabolism, Humans, Jan Yi-Hua, Laskin Debra L, Laskin Jeffrey D, Liver/drug effects/enzymology, Mice, Microsomes, Mishin Vladimir, NEOMED College of Pharmacy, Nitric Oxide Synthase Type II/*antagonists & inhibitors/metabolism, Nitric Oxide/metabolism, Onium Compounds/*pharmacology, Rats, Recombinant Proteins/metabolism, Richardson Jason R, Sprague-Dawley, Szilagyi John T, Time Factors, Toxicological sciences : an official journal of the Society of Toxicology
Reexamining interstitial radiotherapy for PCa.
Tags: *Brachytherapy/adverse effects/instrumentation/methods/trends, *Radioisotopes/adverse effects, 1994, Contemporary urology, Dose-Response Relationship, Forecasting, Humans, Male, Prostatectomy, Prostatic Neoplasms/diagnostic imaging/*radiotherapy, Radiation, Summers J L, Treatment Outcome, Ultrasonography
Sexual dimorphism in vasopressin-induced contraction of rat aorta.
Mesenteric vascular responses to vasopressin during development of DOCA-salt hypertension in male and female rats.
Tags: 1995, 6-Ketoprostaglandin F1 alpha/metabolism, Analysis of Variance, Animals, Arginine Vasopressin/*pharmacology, Blood Pressure/drug effects, Desoxycorticosterone, Dietary, Dinoprostone/metabolism, Dose-Response Relationship, Drug, Female, Hypertension/chemically induced/*physiopathology, In Vitro Techniques, Male, Prostaglandins/analysis/*metabolism, Rats, Reference Values, Sex Characteristics, Sodium, Splanchnic Circulation/drug effects/*physiology, Sprague-Dawley, Stallone J N, The American journal of physiology
Acute and subchronic effects of methylenedioxymethamphetamine [(+/-)MDMA] on locomotion and serotonin syndrome behavior in the rat.
Tags: 1989, 3, 4-methylenedioxyamphetamine, 4-Methylenedioxyamphetamine/analogs & derivatives/*pharmacology, Amphetamines/*pharmacology, Animal/*drug effects, Animals, Behavior, Designer Drugs/*pharmacology, Dose-Response Relationship, Drug, Inbred Strains, Male, Motor Activity/*drug effects, N-Methyl-3, Pharmacology, biochemistry, and behavior, Rats, Receptors, Serotonin/*drug effects, Spanos L J, Time Factors, Yamamoto B K
A comparative analysis of monoaminergic involvement in the spinal antinociceptive action of DAMPGO and DPDPE.
Tags: 1989, 5)-, Ala(2)-MePhe(4)-Gly(5)-, Amines – Physiology, Anesthetics – Pharmacodynamics, Anesthetics/*pharmacology, Animals, Biogenic Monoamines/*physiology, Cell Surface – Drug Effects, Cell Surface – Physiology, Crisp T, D-Penicillamine (2, Dose-Response Relationship, Drug, Enkephalin, Enkephalins, Enkephalins – Pharmacodynamics, Enkephalins/*pharmacology, Inbred Strains, Injections, Intraspinal, Male, Naloxone – Pharmacodynamics, Naloxone/pharmacology, Opioid/drug effects/*physiology, Pain, Pain – Metabolism, Pain/*metabolism, Rats, Receptors, Spanos L J, Spinal, Spinal Cord – Drug Effects, Spinal Cord – Metabolism, Spinal Cord – Physiopathology, Spinal Cord/drug effects/metabolism/*physiopathology, Stafinsky J L
Functional selectivity of NK1 receptor signaling: peptide agonists can preferentially produce receptor activation or desensitization.
Tags: 2006, Animals, CHO Cells, Cricetinae, Dose-Response Relationship, Drug, Humans, Neurokinin-1/agonists/drug effects/*physiology, Rana catesbeiana, Rats, Receptors, Signal Transduction/*physiology, Simmons Mark A, Substance P/metabolism/pharmacology, Tachykinins/metabolism/pharmacology, The Journal of pharmacology and experimental therapeutics
Localization and function of NK(3) subtype tachykinin receptors of layer V pyramidal neurons of the guinea-pig medial prefrontal cortex.
Tags: 2008, Animals, Autoradiography/methods, Dose-Response Relationship, Drug, Drug Interactions, Excitatory Amino Acid Antagonists/pharmacology, Excitatory Postsynaptic Potentials/drug effects/radiation effects, Guinea Pigs, In Vitro Techniques, Iodine Isotopes/pharmacokinetics, Male, Medd A M, Membrane Potentials/drug effects/physiology/radiation effects, Neurokinin B/analogs & derivatives/pharmacokinetics, Neurokinin-3/agonists/antagonists & inhibitors/*metabolism, Neuroscience, Patch-Clamp Techniques, Peptide Fragments/pharmacology, Prefrontal Cortex/*cytology, Protein Binding/drug effects, Pyramidal Cells/drug effects/*metabolism, Quinolines/pharmacology, Quinoxalines/pharmacology, Receptors, Simmons M A, Sobotka-Briner C D, Substance P/analogs & derivatives/pharmacology, Valine/analogs & derivatives/pharmacology
The role of dopamine and serotonin receptors in the mediation of the ethanol interoceptive cue.
Tags: 1988, Animals, Conditioning, Cues, Discrimination (Psychology)/*physiology, Dopamine/drug effects/*physiology, Dose-Response Relationship, Drug, Ethanol/*pharmacology, Inbred Strains, Male, Operant/physiology, Pharmacology, biochemistry, and behavior, Rats, Receptors, Schechter M D, Serotonin/drug effects/*physiology, Signs S A
Stability of the stimulus properties of drugs over time.
Interaction of ethanol and tetrahydro-beta-carboline (THBC) in a discriminative task.
Tags: 1988, Alcohol (Fayetteville, N.Y.), Animal/drug effects, Animals, Behavior, Carbolines/*pharmacology, Conditioning (Psychology)/drug effects, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Drug Interactions, Ethanol/*pharmacology, Inbred Strains, Male, Rats, Schechter M D, Signs S A
Direct microinjection of cathinone into the rat brain produces discriminative stimuli.
Tags: *Brain/anatomy & histology, 1992, Alkaloids/administration & dosage/*pharmacology, Animals, Calcagnetti D J, Discrimination (Psychology)/*drug effects, Discrimination Learning/drug effects, Dose-Response Relationship, Drug, Inbred Strains, Injections, Intraventricular, Male, Microinjections, Nucleus Accumbens/anatomy & histology, Pharmacology, biochemistry, and behavior, Psychotropic Drugs/*pharmacology, Rats, Schechter J B, Schechter M D
Ethanol discrimination in Fawn-Hooded rats is compromised when compared to other strains.
Dopaminergic mediation of the stimulant generalization of nicotine.
Tags: 1993, Alkaloids/pharmacology, Animals, Central Nervous System Stimulants/administration & dosage/*pharmacology, Cues, Discrimination (Psychology)/drug effects, Dopamine/*physiology, Dose-Response Relationship, Drug, Generalization (Psychology)/*drug effects, Injections, Intraperitoneal, Male, Meehan S M, Nicotine/administration & dosage/*pharmacology, Progress in neuro-psychopharmacology & biological psychiatry, Rats, Schechter M D, Sprague-Dawley, Thiazepines/pharmacology
The lethal effects of ethanol and cocaine and their combination in mice: implications for cocaethylene formation.
Tags: 1995, Animals, Central Nervous System Depressants/*toxicity, Cocaine/*analogs & derivatives/metabolism/toxicity, Dopamine Uptake Inhibitors/*toxicity, Dose-Response Relationship, Drug, Drug Interactions, Ethanol/*toxicity, Female, Lethal Dose 50, Male, Meehan S M, Mice, Pharmacology, biochemistry, and behavior, Schechter M D, Sex Characteristics
Further evidence for the mechanisms that may mediate nicotine discrimination.
Tags: 1992, Animals, Calcium Channel Blockers/pharmacology, Dihydropyridines/pharmacology, Discrimination Learning, Dopamine/*metabolism, Dose-Response Relationship, Drug, Inbred Strains, Indoles/pharmacology, Isradipine, Male, Meehan S M, Nicotine/administration & dosage/*pharmacology, Pharmacology, biochemistry, and behavior, Rats, Schechter M D, Thiazepines/pharmacology, Tropisetron
Conditioned place preference produced by the psychostimulant cathinone.
Tags: 1993, Alkaloids/administration & dosage/*pharmacology, Animals, Central Nervous System Stimulants/administration & dosage/*pharmacology, Choice Behavior/drug effects, Conditioning (Psychology)/drug effects, Dose-Response Relationship, Drug, European journal of pharmacology, Habituation, Male, Meehan S M, Motor Activity/*drug effects, Psychophysiologic, Rats, Schechter M D, Sprague-Dawley
Conditioned place aversion produced by dopamine release inhibition.
Tags: 1994, Analysis of Variance, Animal, Animals, Antipsychotic Agents/administration & dosage/*pharmacology, Aversive Therapy, Conditioning (Psychology), Disease Models, Dopamine Antagonists/administration & dosage/*pharmacology, Dose-Response Relationship, Drug, European journal of pharmacology, Injections, Intraperitoneal, Male, Meechan S M, Motor Activity/*drug effects, Random Allocation, Rats, Schechter M D, Sprague-Dawley, Thiazepines/administration & dosage/*pharmacology
Phentermine+fenfluramine produce cocaine-like discriminative cues.
Tags: *Discrimination (Psychology), 1996, Animals, Cocaine/*pharmacology, Department of Anatomy & Neurobiology, Dose-Response Relationship, Drug, Fenfluramine/administration & dosage/*pharmacology, Life sciences, Male, McBurney D, NEOMED College of Medicine, Phentermine/administration & dosage/*pharmacology, Rats, Schechter M D, Sprague-Dawley
Differences in response to the aversive properties and activity effects of low dose ethanol in LAS and HAS selectively bred rats.
Comparison of the behavioral effects of ibogaine from three sources: mediation of discriminative activity.
Lack of generalization of nisoxetine with amphetamine in the rat.
Tags: *Discrimination (Psychology), 1988, Animals, Boja J W, Conditioning, Dextroamphetamine/*pharmacology, Dose-Response Relationship, Drug, Fluoxetine/*analogs & derivatives/pharmacology, Inbred Strains, Male, Norepinephrine/antagonists & inhibitors, Operant/*drug effects, Pharmacology, biochemistry, and behavior, Rats, Reference Values, Schechter M D
CGS 10746B is able to attenuate the effects of amphetamine: further evidence for dopaminergic mediation.
Tags: 1988, Alkaloids/pharmacology, Animals, Antipsychotic Agents/*pharmacology, Apomorphine/pharmacology, Boja J W, Cocaine/pharmacology, Conditioning, Dextroamphetamine/antagonists & inhibitors/*pharmacology, Discrimination (Psychology)/*drug effects, Dopamine/*physiology, Dose-Response Relationship, Drug, Male, Operant/drug effects, Pharmacology, biochemistry, and behavior, Rats, Schechter M D, Thiazepines/*pharmacology
Use of TFMPP stimulus properties as a model of 5-HT1B receptor activation.
Tags: 1988, Animals, Biological, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Male, Models, Norfenfluramine/pharmacology, Pharmaceutical Vehicles, Pharmacology, biochemistry, and behavior, Piperazines/*pharmacology, Rats, Receptors, Schechter M D, Serotonin/*drug effects/physiology, Serotonin/pharmacology
Time-dependent effect of ethanol upon discrimination behavior.
Temporal differences in behavioral effect of fenfluramine and norfenfluramine.
Tags: 1990, Animal/*drug effects, Animals, Behavior, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Fenfluramine/*analogs & derivatives/*pharmacology, Inbred Strains, Injections, Intraperitoneal, Male, Norfenfluramine/*pharmacology, Pharmacology, biochemistry, and behavior, Rats, Schechter M D, Stereoisomerism
Serotonergic-dopaminergic mediation of 3,4-methylenedioxymethamphetamine (MDMA, "ecstasy").
Tags: *Dopamine Antagonists, *Generalization, 1988, 3, 4-methylenedioxyamphetamine, 4-Methylenedioxyamphetamine/analogs & derivatives/*pharmacology, Amphetamines/*pharmacology, Animals, Discrimination (Psychology)/*drug effects, Dopamine Agents/*pharmacology, Dose-Response Relationship, Drug, Inbred Strains, Male, N-Methyl-3, Pharmacology, biochemistry, and behavior, Rats, Schechter M D, Serotonin Antagonists/*pharmacology, Serotonin/*physiology, Stimulus, Time Factors
Rats become acutely tolerant to cathine after amphetamine or cathinone administration.
Tags: 1990, Alkaloids/*pharmacology, Amphetamine/*pharmacology, Animals, Antipsychotic Agents/pharmacology, Discrimination (Psychology)/drug effects, Dose-Response Relationship, Drug, Drug Tolerance, Inbred Strains, Male, Phenylpropanolamine/*pharmacology, Psychopharmacology, Psychotropic Drugs/*pharmacology, Rats, Schechter M D, Thiazepines/pharmacology
Functional consequences of fenfluramine neurotoxicity.
Tags: 1990, Animals, Conditioning, Discrimination Learning/drug effects, Dose-Response Relationship, Drug, Fenfluramine/*toxicity, Inbred Strains, Male, Nervous System Diseases/*chemically induced/psychology, Operant/drug effects, Pharmacology, biochemistry, and behavior, Rats, Reinforcement Schedule, Schechter M D
Effect of MDMA neurotoxicity upon its conditioned place preference and discrimination.
Tags: 1991, 3, 4-methylenedioxyamphetamine, 4-Methylenedioxyamphetamine/*analogs & derivatives/toxicity, Animals, Choice Behavior/*drug effects, Classical/*drug effects, Conditioning, Designer Drugs/*toxicity, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Inbred Strains, Male, N-Methyl-3, Nervous System/*drug effects, Pharmacology, biochemistry, and behavior, Rats, Schechter M D, Sodium Chloride/pharmacology
Dopaminergic nature of acute cathine tolerance.
Tags: 1990, Alkaloids/pharmacology, Animals, Antipsychotic Agents/pharmacology, Appetite Depressants/*pharmacology, Discrimination (Psychology)/drug effects, Discrimination Learning/drug effects, Dopamine/*physiology, Dose-Response Relationship, Drug, Drug Tolerance, Generalization (Psychology)/drug effects, Inbred Strains, Male, Pharmacology, biochemistry, and behavior, Phenylpropanolamine/*pharmacology, Rats, Schechter M D, Thiazepines/pharmacology
Discriminative stimulus effect of phenylephrine.
Tags: 1991, Adrenergic, Adrenergic alpha-Agonists/pharmacology, Adrenergic alpha-Antagonists/pharmacology, alpha/drug effects, Animals, Archives internationales de pharmacodynamie et de therapie, Cues, Discrimination (Psychology)/*drug effects, Dose-Response Relationship, Drug, Generalization, Inbred Strains, Male, Phenylephrine/*pharmacology, Rats, Receptors, Reinforcement Schedule, Schechter M D, Stimulus/drug effects
Comparison of anorectic drugs in rats trained to discriminate between satiation and deprivation.
Tags: *Food Deprivation, 1990, Amphetamine/*pharmacology, Analysis of Variance, Animals, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Fenfluramine/*analogs & derivatives/*pharmacology, Inbred Strains, Life sciences, Male, Norfenfluramine/*pharmacology, Rats, Satiation/*drug effects, Schechter M D