Browse Items (6 total)
- Tags: Tertiary
3D-QSAR and docking studies of pentacycloundecylamines at the sigma-1 (sigma1) receptor.
Tags: *Quantitative Structure-Activity Relationship, 2013, Amines/*chemistry/metabolism, Aza Compounds/chemistry, Binding Sites, Bioorganic & medicinal chemistry letters, Geldenhuys Werner J, Kinetics, Malan Sarel F, Molecular Docking Simulation, Novotny Nicholas, Protein Binding, Protein Structure, Receptors, sigma/*chemistry/metabolism, Tertiary, Van der Schyf Cornelis J
3D-Quantitative structure-activity relationship and docking studies of the tachykinin NK3 receptor.
Tags: *Quantitative Structure-Activity Relationship, 2011, Binding Sites, Bioorganic & medicinal chemistry letters, Computer Simulation, Drug Design, Geldenhuys Werner J, Humans, Ligands, Models, Molecular, Neurokinin-3/*chemistry/metabolism, Protein Structure, Quinolines/chemistry, Receptors, Simmons Mark A, Tertiary
A Prospero-related homeodomain protein is a novel co-regulator of hepatocyte nuclear factor 4alpha that regulates the cholesterol 7alpha-hydroxylase gene.
Tags: *Gene Expression Regulation, 2006, Aged, Amino Acid Motifs, Bile Acids and Salts/metabolism, Cell Line, Cell Nucleus/metabolism, Cells, Chiang John Y L, Cholesterol 7-alpha-Hydroxylase/*chemistry/*genetics, Cultured/metabolism, Department of Integrative Medical Sciences, Enzymologic, Female, Genes, Genetic, Gluconeogenesis, Glutathione Transferase/metabolism, Hepatocyte Nuclear Factor 4/metabolism/*physiology, Hepatocytes/metabolism, Homeodomain Proteins/metabolism/*physiology, Humans, Immunoprecipitation, Li Tiangang, Liver/metabolism, Luciferases/metabolism, Male, Messenger/metabolism, Middle Aged, NEOMED College of Medicine, Phosphoenolpyruvate Carboxykinase (ATP)/metabolism, Plasmids/metabolism, Protein Structure, Reporter, Response Elements, Reverse Transcriptase Polymerase Chain Reaction, RNA, Small Interfering/metabolism, Song Kwang-Hoon, Tertiary, The Journal of biological chemistry, Time Factors, Transcription, Transcriptional Activation, Transfection, Tumor Suppressor Proteins, Two-Hybrid System Techniques
Design and use of peptide-based antibodies decreasing superoxide production by mitochondrial complex I and complex II.
Tags: *Electron Transport Complex I/antagonists & inhibitors/chemistry/immunology/metabolism, *Electron Transport Complex II/antagonists & inhibitors/chemistry/immunology/metabolism, *Mitochondria, *Mitochondrial Proteins/antagonists & inhibitors/chemistry/immunology/metabolism, *Peptides/chemistry/immunology/metabolism, 2011, Amino Acid Motifs, Animals, Biopolymers, Cattle, Chen Yeong-Renn, Department of Integrative Medical Sciences, Female, Heart/chemistry/immunology/metabolism, Kang Patrick T, Kaumaya Pravin P T, NEOMED College of Medicine, Protein Structure, Rabbits, Tertiary, Yun June
Inhibition of monoamine oxidase by derivatives of piperine, an alkaloid from the pepper plant Piper nigrum, for possible use in Parkinson's disease.
Tags: 2012, Al-Baghdadi Osamah B, Alkaloids/*chemistry/isolation & purification/pharmacology, Animals, Benzodioxoles/*chemistry/isolation & purification/pharmacology, Binding Sites, Bioorganic & medicinal chemistry letters, Blood-Brain Barrier/drug effects, Bovine/metabolism, Cattle, Geldenhuys Werner J, Humans, Hydrogen Bonding, Molecular Docking Simulation, Monoamine Oxidase Inhibitors/*chemistry/isolation & purification/pharmacology, Monoamine Oxidase/*chemistry/metabolism, Parkinson Disease/metabolism/pathology, Piper nigrum/*chemistry, Piperidines/*chemistry/isolation & purification/pharmacology, Polyunsaturated Alkamides/*chemistry/isolation & purification/pharmacology, Prater Natalie I, Protein Binding, Protein Structure, Serum Albumin, Tertiary, Van der Schyf Cornelis J
Novel compounds that target lipoprotein lipase and mediate growth arrest in acute lymphoblastic leukemia.
Tags: *Acute lymphoblastic leukemia, *Cancer, *Co-culture model, *Lipids, *Lipoprotein lipase, *Metabolism, 2018, Amides/chemistry/metabolism/pharmacology, Antineoplastic Agents/*chemistry/metabolism/pharmacology, Binding Sites, Bioorganic & medicinal chemistry letters, Cell Line, Cell Proliferation/drug effects, Coculture Techniques, Department of Pharmaceutical Sciences, Department of Pharmacy Practice, Dyslipidemias/complications/metabolism/pathology, Geldenhuys Werner J, Gibson Laura F, Humans, Lipoprotein Lipase/antagonists & inhibitors/*metabolism, Mesenchymal Stem Cells/cytology/metabolism, Molecular Docking Simulation, Nair Rajesh R, NEOMED College of Graduate Studies, NEOMED College of Pharmacy, Piktel Debbie, Precursor Cell Lymphoblastic Leukemia-Lymphoma/complications/metabolism/pathology, Protein Binding, Protein Structure, Sadana Prabodh, Serum Albumin/chemistry/metabolism, Tertiary, Tumor