Browse Items (132 total)
- Tags: Dose-Response Relationship
Clinical impact of temporary therapy interruptions on anticoagulation control in patients treated with warfarin.
Tags: 2013, Aged, American journal of therapeutics, Anticoagulants – Administration and Dosage, Anticoagulants – Therapeutic Use, Atrial Fibrillation – Drug Therapy, Blood Coagulation Disorders – Drug Therapy, Boros Melanie L, Coronary Thrombosis – Drug Therapy, Department of Pharmaceutical Sciences, Department of Pharmacy Practice, Dose-Response Relationship, Drug, Drug Administration Schedule, Drug Monitoring, Euthanasia, Female, Gallegos Patrick J, Human, International Normalized Ratio, Male, Middle Age, NEOMED College of Pharmacy, Passive, Postoperative Care, Preoperative Care, Prospective Studies, Retrospective Design, Rybarczyk Amy M, Treatment Outcomes, Venous Thromboembolism – Drug Therapy, Warfarin – Administration and Dosage, Warfarin – Therapeutic Use, Zimmerman Jacob P
Efficacy of Higher-dose Oseltamivir in Adults with Influenza A and B.
Tags: 2014, Department of Internal Medicine, Dose-Response Relationship, Infectious Disease Alert, Influenza A Virus, Influenza – Drug Therapy, Influenza B Virus, Multicenter Studies, NEOMED College of Medicine, Oseltamivir – Adverse Effects, Oseltamivir – Therapeutic Use, Prospective Studies, Treatment Outcomes, Watkins Richard R
Steroids Increase the Risk for Community-acquired Staphylococcus aureus Bacteremia...Smit J, Kaasch AJ, Sogaard M , t al. Use of glucocorticoids and risk of community-acquired Staphylococcus aureus bacteremia:A population-based case-control study. Mayo Clin Proc 2016 :91:873-880.
Tags: 2016, Bacteremia – Risk Factors, Community-Acquired Infections – Risk Factors, Denmark, Department of Internal Medicine, Dose-Response Relationship, Drug, Glucocorticoids – Adverse Effects, Infectious Disease Alert, NEOMED College of Medicine, Staphylococcal Infections – Risk Factors, Staphylococcus aureus, Watkins Richard R
Reexamining interstitial radiotherapy for PCa.
Tags: *Brachytherapy/adverse effects/instrumentation/methods/trends, *Radioisotopes/adverse effects, 1994, Contemporary urology, Dose-Response Relationship, Forecasting, Humans, Male, Prostatectomy, Prostatic Neoplasms/diagnostic imaging/*radiotherapy, Radiation, Summers J L, Treatment Outcome, Ultrasonography
A comparative analysis of monoaminergic involvement in the spinal antinociceptive action of DAMPGO and DPDPE.
Tags: 1989, 5)-, Ala(2)-MePhe(4)-Gly(5)-, Amines – Physiology, Anesthetics – Pharmacodynamics, Anesthetics/*pharmacology, Animals, Biogenic Monoamines/*physiology, Cell Surface – Drug Effects, Cell Surface – Physiology, Crisp T, D-Penicillamine (2, Dose-Response Relationship, Drug, Enkephalin, Enkephalins, Enkephalins – Pharmacodynamics, Enkephalins/*pharmacology, Inbred Strains, Injections, Intraspinal, Male, Naloxone – Pharmacodynamics, Naloxone/pharmacology, Opioid/drug effects/*physiology, Pain, Pain – Metabolism, Pain/*metabolism, Rats, Receptors, Spanos L J, Spinal, Spinal Cord – Drug Effects, Spinal Cord – Metabolism, Spinal Cord – Physiopathology, Spinal Cord/drug effects/metabolism/*physiopathology, Stafinsky J L
Acute and subchronic effects of methylenedioxymethamphetamine [(+/-)MDMA] on locomotion and serotonin syndrome behavior in the rat.
Tags: 1989, 3, 4-methylenedioxyamphetamine, 4-Methylenedioxyamphetamine/analogs & derivatives/*pharmacology, Amphetamines/*pharmacology, Animal/*drug effects, Animals, Behavior, Designer Drugs/*pharmacology, Dose-Response Relationship, Drug, Inbred Strains, Male, Motor Activity/*drug effects, N-Methyl-3, Pharmacology, biochemistry, and behavior, Rats, Receptors, Serotonin/*drug effects, Spanos L J, Time Factors, Yamamoto B K
The role of dopamine and serotonin receptors in the mediation of the ethanol interoceptive cue.
Tags: 1988, Animals, Conditioning, Cues, Discrimination (Psychology)/*physiology, Dopamine/drug effects/*physiology, Dose-Response Relationship, Drug, Ethanol/*pharmacology, Inbred Strains, Male, Operant/physiology, Pharmacology, biochemistry, and behavior, Rats, Receptors, Schechter M D, Serotonin/drug effects/*physiology, Signs S A
Use of TFMPP stimulus properties as a model of 5-HT1B receptor activation.
Tags: 1988, Animals, Biological, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Male, Models, Norfenfluramine/pharmacology, Pharmaceutical Vehicles, Pharmacology, biochemistry, and behavior, Piperazines/*pharmacology, Rats, Receptors, Schechter M D, Serotonin/*drug effects/physiology, Serotonin/pharmacology
Time-dependent effect of ethanol upon discrimination behavior.
Temporal differences in behavioral effect of fenfluramine and norfenfluramine.
Tags: 1990, Animal/*drug effects, Animals, Behavior, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Fenfluramine/*analogs & derivatives/*pharmacology, Inbred Strains, Injections, Intraperitoneal, Male, Norfenfluramine/*pharmacology, Pharmacology, biochemistry, and behavior, Rats, Schechter M D, Stereoisomerism
Stability of the stimulus properties of drugs over time.
Serotonergic-dopaminergic mediation of 3,4-methylenedioxymethamphetamine (MDMA, "ecstasy").
Tags: *Dopamine Antagonists, *Generalization, 1988, 3, 4-methylenedioxyamphetamine, 4-Methylenedioxyamphetamine/analogs & derivatives/*pharmacology, Amphetamines/*pharmacology, Animals, Discrimination (Psychology)/*drug effects, Dopamine Agents/*pharmacology, Dose-Response Relationship, Drug, Inbred Strains, Male, N-Methyl-3, Pharmacology, biochemistry, and behavior, Rats, Schechter M D, Serotonin Antagonists/*pharmacology, Serotonin/*physiology, Stimulus, Time Factors
Rats become acutely tolerant to cathine after amphetamine or cathinone administration.
Tags: 1990, Alkaloids/*pharmacology, Amphetamine/*pharmacology, Animals, Antipsychotic Agents/pharmacology, Discrimination (Psychology)/drug effects, Dose-Response Relationship, Drug, Drug Tolerance, Inbred Strains, Male, Phenylpropanolamine/*pharmacology, Psychopharmacology, Psychotropic Drugs/*pharmacology, Rats, Schechter M D, Thiazepines/pharmacology
Lack of generalization of nisoxetine with amphetamine in the rat.
Tags: *Discrimination (Psychology), 1988, Animals, Boja J W, Conditioning, Dextroamphetamine/*pharmacology, Dose-Response Relationship, Drug, Fluoxetine/*analogs & derivatives/pharmacology, Inbred Strains, Male, Norepinephrine/antagonists & inhibitors, Operant/*drug effects, Pharmacology, biochemistry, and behavior, Rats, Reference Values, Schechter M D
Interaction of ethanol and tetrahydro-beta-carboline (THBC) in a discriminative task.
Tags: 1988, Alcohol (Fayetteville, N.Y.), Animal/drug effects, Animals, Behavior, Carbolines/*pharmacology, Conditioning (Psychology)/drug effects, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Drug Interactions, Ethanol/*pharmacology, Inbred Strains, Male, Rats, Schechter M D, Signs S A
Functional consequences of fenfluramine neurotoxicity.
Tags: 1990, Animals, Conditioning, Discrimination Learning/drug effects, Dose-Response Relationship, Drug, Fenfluramine/*toxicity, Inbred Strains, Male, Nervous System Diseases/*chemically induced/psychology, Operant/drug effects, Pharmacology, biochemistry, and behavior, Rats, Reinforcement Schedule, Schechter M D
Effect of MDMA neurotoxicity upon its conditioned place preference and discrimination.
Tags: 1991, 3, 4-methylenedioxyamphetamine, 4-Methylenedioxyamphetamine/*analogs & derivatives/toxicity, Animals, Choice Behavior/*drug effects, Classical/*drug effects, Conditioning, Designer Drugs/*toxicity, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Inbred Strains, Male, N-Methyl-3, Nervous System/*drug effects, Pharmacology, biochemistry, and behavior, Rats, Schechter M D, Sodium Chloride/pharmacology
Dopaminergic nature of acute cathine tolerance.
Tags: 1990, Alkaloids/pharmacology, Animals, Antipsychotic Agents/pharmacology, Appetite Depressants/*pharmacology, Discrimination (Psychology)/drug effects, Discrimination Learning/drug effects, Dopamine/*physiology, Dose-Response Relationship, Drug, Drug Tolerance, Generalization (Psychology)/drug effects, Inbred Strains, Male, Pharmacology, biochemistry, and behavior, Phenylpropanolamine/*pharmacology, Rats, Schechter M D, Thiazepines/pharmacology
Discriminative stimulus effect of phenylephrine.
Tags: 1991, Adrenergic, Adrenergic alpha-Agonists/pharmacology, Adrenergic alpha-Antagonists/pharmacology, alpha/drug effects, Animals, Archives internationales de pharmacodynamie et de therapie, Cues, Discrimination (Psychology)/*drug effects, Dose-Response Relationship, Drug, Generalization, Inbred Strains, Male, Phenylephrine/*pharmacology, Rats, Receptors, Reinforcement Schedule, Schechter M D, Stimulus/drug effects
Comparison of anorectic drugs in rats trained to discriminate between satiation and deprivation.
Tags: *Food Deprivation, 1990, Amphetamine/*pharmacology, Analysis of Variance, Animals, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Fenfluramine/*analogs & derivatives/*pharmacology, Inbred Strains, Life sciences, Male, Norfenfluramine/*pharmacology, Rats, Satiation/*drug effects, Schechter M D
CGS 10746B is able to attenuate the effects of amphetamine: further evidence for dopaminergic mediation.
Tags: 1988, Alkaloids/pharmacology, Animals, Antipsychotic Agents/*pharmacology, Apomorphine/pharmacology, Boja J W, Cocaine/pharmacology, Conditioning, Dextroamphetamine/antagonists & inhibitors/*pharmacology, Discrimination (Psychology)/*drug effects, Dopamine/*physiology, Dose-Response Relationship, Drug, Male, Operant/drug effects, Pharmacology, biochemistry, and behavior, Rats, Schechter M D, Thiazepines/*pharmacology
Advantages and disadvantages of a rapid method to train drug discrimination.
Tags: 1988, 3, 4-methylenedioxyamphetamine, 4-Methylenedioxyamphetamine/analogs & derivatives/*pharmacology, Amphetamines/*pharmacology, Animals, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Drug Tolerance, Male, Methods, N-Methyl-3, Pharmacology, biochemistry, and behavior, Rats, Schechter M D
Guggulsterone antagonizes farnesoid X receptor induction of bile salt export pump but activates pregnane X receptor to inhibit cholesterol 7alpha-hydroxylase gene.
Tags: 2003, ATP Binding Cassette Transporter, ATP-Binding Cassette Transporters/*genetics, Biochemical and biophysical research communications, Cell Line, Chenodeoxycholic Acid/antagonists & inhibitors, Chiang John Y L, Cholesterol 7-alpha-Hydroxylase/*genetics, Cytoplasmic and Nuclear/*metabolism, Department of Integrative Medical Sciences, DNA-Binding Proteins/*antagonists & inhibitors/metabolism, Dose-Response Relationship, Drug, Gene Expression Regulation/drug effects, Humans, Member 11, NEOMED College of Medicine, Owsley Erika, Pregnane X Receptor, Pregnenediones/*pharmacology, Receptors, Steroid/*metabolism, Subfamily B, Transcription Factors/*antagonists & inhibitors/metabolism, Transcriptional Activation/drug effects
Inverse agonist properties of the FG 7142 discriminative stimulus.
Tags: 1991, Animals, Appetite Depressants/*pharmacology, Carbolines/antagonists & inhibitors/*pharmacology, Discrimination (Psychology)/*drug effects, Discrimination Learning/drug effects, Dose-Response Relationship, Drug, GABA-A/drug effects, Generalization, Inbred Strains, Leidenheimer N J, Male, Pharmacology, biochemistry, and behavior, Rats, Receptors, Reinforcement Schedule, Schechter M D, Stimulus/drug effects
Inverse agonist properties of the THBC discriminative stimulus: asymmetrical generalization with FG 7142.
Tags: 1991, Animals, Avoidance Learning/drug effects, Carbolines/antagonists & inhibitors/*pharmacology, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, GABA-A/*drug effects, Generalization, Inbred Strains, Leidenheimer N J, Male, Pharmacology, biochemistry, and behavior, Rats, Receptors, Schechter M D, Stimulus/*drug effects
Discriminative stimulus properties of CGS 9896: interactions within the GABA/benzodiazepine receptor complex.
Tags: 1988, Animals, Carbolines/pharmacology, Chlordiazepoxide/pharmacology, Discrimination (Psychology)/drug effects/*physiology, Dose-Response Relationship, Drug, Flumazenil/pharmacology, GABA-A/*physiology, gamma-Aminobutyric Acid/analogs & derivatives/pharmacology, Inbred Strains, Leidenheimer N J, Male, Pentobarbital/pharmacology, Pentylenetetrazole/pharmacology, Pharmacology, biochemistry, and behavior, Pyrazoles/antagonists & inhibitors/*metabolism, Rats, Receptors, Schechter M D
Time and dose dependency of the suppression of pulmonary metastases of rat mammary cancer by amiloride.
Tags: 1998, Amiloride/*administration & dosage, Animals, Antineoplastic Agents/*administration & dosage, Arvan M, Clinical & experimental metastasis, Dose-Response Relationship, Drug, Drug Administration Schedule, Evans D M, Experimental/*pathology, Female, Guyton D P, Inbred F344, Lung Neoplasms/pathology/*prevention & control/*secondary, Mammary Neoplasms, Neoplasm Transplantation, Plasminogen Activators/antagonists & inhibitors, Rats, Sloan-Stakleff K, Urokinase-Type Plasminogen Activator/antagonists & inhibitors
The antinociceptive effects of 3,4-methylenedioxymethamphetamine (MDMA) in the rat.
Tags: 1989, 3, 4-methylenedioxyamphetamine, 4-Methylenedioxyamphetamine/analogs & derivatives/*pharmacology, Amphetamines/*pharmacology, Analgesics/*pharmacology, Animals, Boja J W, Crisp T, Dose-Response Relationship, Drug, Inbred Strains, Male, Methysergide/pharmacology, Morphine/pharmacology, N-Methyl-3, Naltrexone/pharmacology, Pain/*metabolism, Pharmacology, biochemistry, and behavior, Rats, Receptors, Schechter M D, Serotonin/drug effects/*physiology, Stafinsky J L
Age-related changes in the spinal antinociceptive effects of DAGO, DPDPE and beta-endorphin in the rat.
Tags: 1994, 5)-, Aging/*physiology, Ala(2)-MePhe(4)-Gly(5)-, Analgesics/*pharmacology, Analysis of Variance, Animals, beta-Endorphin/administration & dosage/*pharmacology, Brain research, Crisp T, D-Penicillamine (2, Dose-Response Relationship, Drug, Enkephalin, Enkephalins/administration & dosage/*pharmacology, Gordon T L, Hoskins D L, Inbred F344, Injections, Male, Pain/*physiopathology, Perni V C, Rats, Spinal, Spine/drug effects/growth & development/*physiology, Stafinsky J L, Uram M
Testosterone causes direct relaxation of rat thoracic aorta.
Tags: 1996, Animals, Aorta, Calcium Channels/drug effects, Costarella C E, Department of Internal Medicine, Dose-Response Relationship, Drug, Endothelium, Female, In Vitro Techniques, Male, NEOMED College of Medicine, Phenylephrine/pharmacology, Rats, Rutecki G W, Sprague-Dawley, Stallone J N, Testosterone/*pharmacology, The Journal of pharmacology and experimental therapeutics, Thoracic/*drug effects/physiology, Vascular/physiology, Vasodilation/*drug effects, Whittier F C
Regulation of human sterol 27-hydroxylase gene (CYP27A1) by bile acids and hepatocyte nuclear factor 4alpha (HNF4alpha).
Tags: *DNA-Binding Proteins, 2003, Base Sequence, Basic Helix-Loop-Helix Leucine Zipper Transcription Factors, Bile Acids and Salts/*pharmacology, Binding Sites/genetics, Cell Line, Chen Wenling, Chenodeoxycholic Acid/pharmacology, Chiang John Y L, Cholestanetriol 26-Monooxygenase, Cloning, Cultured, Cytoplasmic and Nuclear/genetics/metabolism, Department of Integrative Medical Sciences, DNA, DNA/chemistry/genetics, Dose-Response Relationship, Drug, gene, Gene Expression Regulation/drug effects, Genetic/*genetics, Hepatocyte Nuclear Factor 4, Humans, Luciferases/genetics/metabolism, Molecular, Molecular Sequence Data, Mutagenesis, Mutation, NEOMED College of Medicine, Phosphoproteins/genetics/*metabolism, Promoter Regions, Receptors, Recombinant Fusion Proteins/genetics/metabolism, Response Elements/genetics, Sequence Analysis, Site-Directed, Steroid Hydroxylases/*genetics, Transcription Factors/genetics/*metabolism, Transfection, Tumor Cells
Norfenfluramine, the fenfluramine metabolite, provides stimulus control: evidence for serotonergic mediation.
Tags: 1988, Animal/*drug effects, Animals, Behavior, Boja J W, Discrimination (Psychology)/*drug effects, Dose-Response Relationship, Drug, Fenfluramine/*analogs & derivatives/*pharmacology, Inbred Strains, Male, Norfenfluramine/*pharmacology, Pharmacology, biochemistry, and behavior, Rats, Receptors, Schechter M D, Serotonin/pharmacology, Serotonin/physiology, Time Factors
Increased drug sensitivity in the drug discrimination procedure afforded by drug versus drug training.
Tags: 1990, Amphetamine/pharmacology, Animals, Boja J W, Discrimination (Psychology)/*drug effects, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Inbred Strains, Male, Norfenfluramine/pharmacology, Pentobarbital/pharmacology, Psychopharmacology, Rats, Reinforcement Schedule, Schechter M D
Behavioral effects of N-ethyl-3,4-methylenedioxyamphetamine (MDE; "EVE").
Tags: 1987, 3, 4-methylenedioxyamphetamine, 4-Methylenedioxyamphetamine/analogs & derivatives/*pharmacology, Amphetamines/*pharmacology, Animals, Boja J W, Discrimination (Psychology), Dose-Response Relationship, Drug, Inbred Strains, Legislation, Male, N-Methyl-3, Pharmacology, biochemistry, and behavior, Rats, Schechter M D, Time Factors, United States
Time-dependent changes in norepinephrine-induced left ventricular dysfunction and histopathologic condition.
Tags: 1998, Allman F D, Animals, Bosso F J, Dose-Response Relationship, Drug, Female, Herold W, Left/*chemically induced/pathology, Left/drug effects, Male, Myocardial Contraction/drug effects, Myocardial Infarction/chemically induced/pathology, Myocardium/pathology, Norepinephrine/*toxicity, Pilati C F, Rabbits, Systole/drug effects/physiology, The Journal of heart and lung transplantation : the official publication of the International Society for Heart Transplantation, Ventricular Dysfunction, Ventricular Function
Anti-Inflammatory Mechanism Involved in Pomegranate-Mediated Prevention of Breast Cancer: the Role of NF-kappaB and Nrf2 Signaling Pathways.
Tags: 10-Dimethyl-1, 2-benzanthracene/toxicity, 2017, 9, Animal Studies, Animals, Anti-Inflammatory Agents/*pharmacology, anti-inflammatory effects, Anticarcinogenic Agents/pharmacology, Apoptosis/drug effects, Bhatia Deepak, Bishayee Anupam, Breast Neoplasms, breast tumor, Cell Transformation, Chemoprevention, COX-2, Cyclooxygenase 2/genetics/metabolism, DMBA, Dose-Response Relationship, Drug, Experimental/*prevention & control, Female, Gene Expression Regulation, HSP90, HSP90 Heat-Shock Proteins/genetics/metabolism, I-kappa B Kinase/genetics/metabolism, Inflammation Mediators, Mammary Neoplasms, Mandal Animesh, Neoplasms – Prevention and Control, Neoplastic, Neoplastic/drug effects, NF-E2-Related Factor 2/genetics/*metabolism, NF-kappa B/genetics/*metabolism, NF-kappaB, Nrf2, Nutrients, Physical Education and Training, Plant Preparations/*pharmacology, Pomegranate, Punica granatum, Punicaceae/*chemistry, Rats, Signal Transduction
Persistent left ventricular dysfunction after cocaine treatment in rabbits.
Tags: 1993, Anesthesia, Animals, Blood Pressure/drug effects, Cocaine/*pharmacology, Consciousness, Dose-Response Relationship, Drug, Epinephrine/blood, Espinal A R, Female, General, Heart/drug effects/physiology/*physiopathology, In Vitro Techniques, Left/*drug effects, Male, Norepinephrine/blood, Pilati C F, Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), Pukys T F, Rabbits, Stroke Volume/drug effects, Ventricular Function
Antitumor activities of extracts from selected desert plants against HepG2 human hepatocellular carcinoma cells.
Tags: 2013, Aerial, Antineoplastic Agents, Bishayee Anupam, Carcinoma, Desert Climate, Dose-Response Relationship, Drug, Harlev Eli, Hep G2 Cells, Hepatocellular/*drug therapy/pathology, Humans, Inhibitory Concentration 50, Liver Neoplasms/*drug therapy/pathology, Mandal Animesh, Medicinal/chemistry, Nevo Eviatar, Pharmaceutical biology, Phytogenic/administration & dosage/*pharmacology, Plant Components, Plant Extracts/administration & dosage/*pharmacology, Plants, Tetrazolium Salts/chemistry, Thiazoles/chemistry, Thoppil Roslin J, Time Factors
Solutions to the problem of bacterial resistance.
Tags: *Drug Resistance, *Practice Guidelines as Topic, 2005, Anti-Bacterial Agents/*therapeutic use, Bacterial, Department of Internal Medicine, Dose-Response Relationship, Drug, Drug Administration Schedule, Drug Prescriptions/standards, Drug Utilization, File Thomas M Jr, Humans, NEOMED College of Medicine, Professional Practice/*standards, Treatments in respiratory medicine, Unnecessary Procedures