Browse Items (27 total)
- Tags: Kinetics
Use of in vitro superfusion to assess the dynamics of striatal dopamine clearance: influence of estrogen.
The modulation of long-term potentiation by delta-9-tetrahydrocannabinol in the rat hippocampus, in vitro.
Stabilization of clathrin coated vesicles by amantadine, tromantadine and other hydrophobic amines.
Relationships between Very Low-Density Lipoproteins-Ceramides, -Diacylglycerols, and -Triacylglycerols in Insulin-Resistant Men.
Tags: 2020, Biomarkers, Ceramides, Department of Pharmaceutical Sciences, Disease, Gaballah Ayman, Garrett Timothy J, Humans, Inflammation, journalArticle, June 2020 Update II, Kasumov Takhar, Kinetics, LDL, Lipids, Manrique-Acevedo Camila, Metabolic syndrome, Mucinski Justine M, NAFLD, NEOMED College of Pharmacy, obese men, Parks Elizabeth J, secretion, sphingolipids, VLDL
Regulation of cholesterol 7 alpha-hydroxylase in the liver. Purification of cholesterol 7 alpha-hydroxylase and the immunochemical evidence for the induction of cholesterol 7 alpha-hydroxylase by cholestyramine and circadian rhythm.
Tags: *Circadian Rhythm, 1990, Animals, Chiang J Y, Cholesterol 7-alpha-Hydroxylase/*biosynthesis/isolation & purification/metabolism, Cholestyramine Resin/*pharmacology, Chromatography, Department of Integrative Medical Sciences, Durapatite, Enzyme Induction, Hydroxyapatites, Inbred Strains, Ion Exchange, Isoenzymes/*biosynthesis/isolation & purification, Kinetics, Lin G M, Liver/drug effects/*enzymology, Microsomes, Miller W F, NEOMED College of Medicine, Obesity/enzymology, Organ Specificity, Polyethylene Glycols, Rats, Steroid Hydroxylases/*biosynthesis, The Journal of biological chemistry, Zucker
Regulation of cholesterol 7 alpha-hydroxylase in the liver. Cloning, sequencing, and regulation of cholesterol 7 alpha-hydroxylase mRNA.
Tags: *Gene Expression Regulation, 1990, Amino Acid Sequence, Animals, Base Sequence, Cell Fractionation, Centrifugation, Chiang J Y, Cholesterol 7-alpha-Hydroxylase/biosynthesis/*genetics/immunology, Cholestyramine Resin/pharmacology, Circadian Rhythm, Cloning, Cytochrome P-450 Enzyme System/genetics, Density Gradient, Department of Integrative Medical Sciences, DNA/genetics/isolation & purification, Enzyme Induction, Enzymologic, Epitopes/analysis, Female, Immunoblotting, Inbred Strains, Kinetics, Li Y C, Liver/drug effects/*enzymology, Messenger/*genetics, Molecular Sequence Data, Molecular/methods, NEOMED College of Medicine, Nucleic Acid, Polyribosomes/metabolism/ultrastructure, Rats, Restriction Mapping, RNA, Sequence Homology, Steroid Hydroxylases/*genetics, The Journal of biological chemistry, Wang D P
Quinone and nitrofurantoin redox cycling by recombinant cytochrome b5 reductase.
Tags: *Cytochrome b5, *Free radicals, *Reactive oxygen species, *redox cycling, 2018, Aleksunes Lauren M, Benzoquinones/*metabolism, Cytochrome-B(5) Reductase/*metabolism, Free Radicals/metabolism, Fussell Karma C, Heck Diane E, Humans, Jan Yi-Hua, Kinetics, Laskin Debra L, Laskin Jeffrey D, Liver, Microsomes, Mishin Vladimir, NADP/metabolism, Nitrofurantoin/*metabolism, Oxidation-Reduction, Oxygen Consumption, Reactive Oxygen Species/metabolism, Recombinant Proteins/metabolism, Richardson Jason R, Szilagyi John T, Toxicology and applied pharmacology, Wang Yun, Yang Shaojun
Quantifying ceramide kinetics in vivo using stable isotope tracers and LC-MS/MS.
Tags: 2018, American journal of physiology. Endocrinology and metabolism, Berejnaia Olga, Chen Ying, Daurio Natalie A, Department of Pharmaceutical Sciences, dyslipidemia, Insulin Resistance, Kasumov Takhar, Kelley David E, Kinetics, lipid turnover, Liu Jinqi, Mass spectrometry, Mayoral Rafael, McLaren David G, NEOMED College of Pharmacy, Petrov Aleksandr, Previs Stephen F, Wang Sheng-Ping, Yin Wu, Zhang Guo-Fang
Prostate apoptosis response-4 enhances secretion of amyloid beta peptide 1-42 in human neuroblastoma IMR-32 cells by a caspase-dependent pathway.
Tags: *Intracellular Signaling Peptides and Proteins, 2001, Amyloid beta-Peptides/*biosynthesis/metabolism, Apoptosis Regulatory Proteins, Apoptosis/*physiology, Carrier Proteins/genetics/*physiology, Caspases/*metabolism, Chang X, Cultured, Du H, Enzyme Activation, Guo Q, Humans, Kinetics, Leucine Zippers, Neuroblastoma, Peptide Fragments/*biosynthesis/metabolism, Recombinant Proteins/metabolism, The Journal of biological chemistry, Time Factors, Transfection, Tumor Cells, Xie J
Pregnancy zone protein is a carrier and modulator of placental protein-14 in
Tags: 2004, alpha-Macroglobulins/immunology/metabolism, Antigens, Carrier Proteins/immunology/metabolism/*physiology, CD/drug effects/immunology, Cell Proliferation/drug effects, Cellular immunology, Cytokines/*biosynthesis/drug effects, Female, Glycodelin, Glycoproteins/immunology/metabolism/*physiology, Humans, Interleukin-2/biosynthesis, Interleukin-4/biosynthesis, Kinetics, Kiyatkina Nadya, Koo Peter H, LEUKOCYTES, Low Density Lipoprotein Receptor-Related Protein-1, Lymphocyte Activation/immunology, Mononuclear/drug effects/immunology, Pregnancy, Pregnancy Proteins/immunology/metabolism/*physiology, Protein Binding, Skornicka Erin L, T-Lymphocytes/cytology/drug effects/*immunology, Time Factors, Tykocinski Mark L, Weber Matthew C
Multiple binding sites for [125I]RTI-121 and other cocaine analogs in rat frontal cerebral cortex.
Tags: *Membrane Transport Proteins, *Nerve Tissue Proteins, *Symporters, 1998, Animals, Binding, Binding Sites, Boja J W, Carrier Proteins/*metabolism, Carroll F I, Cocaine/*analogs & derivatives/pharmacokinetics, Competitive, Corpus Striatum/*metabolism, Dopamine Plasma Membrane Transport Proteins, Dopamine/metabolism, Frontal Lobe/*metabolism, Iodine Radioisotopes/*pharmacokinetics, Kinetics, Kopajtic T, Kuhar M J, Male, Membrane Glycoproteins/*metabolism, Norepinephrine Plasma Membrane Transport Proteins, Norepinephrine/metabolism, Rats, Regression Analysis, Serotonin Plasma Membrane Transport Proteins, Serotonin/metabolism, Sprague-Dawley, Synapse (New York, N.Y.), Vaughan R A
Monitoring the synthesis of biomolecules using mass spectrometry.
Tags: 2016, biosynthesis, Department of Pharmaceutical Sciences, Deuterium Oxide/chemistry, deuterium water, flux analysis, Kasumov Takhar, Kinetics, Macromolecular Substances/*chemistry/*metabolism, Mass spectrometry, Mass Spectrometry/*methods, Metabolomics, Miyagi Masaru, NEOMED College of Pharmacy, Philosophical transactions. Series A, Mathematical, physical, and engineering sciences, proteomics
Mice transgenic for simian immunodeficiency virus nef are immunologically compromised.
Tags: *Genes, *Herpesvirus 1, *Immunocompromised Host, 1998, 3T3 Cells, Aging, Animals, Antibodies, Antibody Formation, Cellular, Cercopithecus aethiops, Docherty J J, Female, Herpes Simplex/*immunology, HIV/pathogenicity, Human, Humans, Immunity, Immunoglobulin G/blood, Journal of biomedical science, Kestler H W, Kinetics, Larsen N B, Male, Mice, nef, Simian Immunodeficiency Virus/*genetics/pathogenicity, Transgenic, Vero Cells, Viral/biosynthesis/blood
Inhibition of rat brain pyruvate dehydrogenase by thiamine analogs.
Tags: 1988, Animals, Biochemical pharmacology, Brain/*enzymology, Cerebral Cortex/drug effects/enzymology, Hippocampus/drug effects/enzymology, Inbred Strains, Kandiko C T, Kinetics, Male, Pyruvate Dehydrogenase Complex/*antagonists & inhibitors, Rats, Smith D, Thiamine Pyrophosphate/analogs & derivatives/pharmacology, Thiamine/*analogs & derivatives/pharmacology, Yamamoto B K
Hyperpolarizing and depolarizing GABAA receptor-mediated dendritic inhibition in area CA1 of the rat hippocampus.
Tags: 1991, 2-Amino-5-phosphonovalerate/pharmacology, Animals, Bicuculline/analogs & derivatives/pharmacology, Borroni A M, Chlorides/pharmacology, Dendrites/drug effects/*physiology, Evoked Potentials/drug effects, GABA-A Receptor Antagonists, GABA-A/drug effects/*physiology, Grover L M, Hippocampus/*physiology, In Vitro Techniques, Journal of neurophysiology, Kinetics, Lambert N A, Mathematics, Membrane Potentials/drug effects, Models, Neurological, Neurons/drug effects/*physiology, Organophosphorus Compounds/pharmacology, Pyramidal Tracts/drug effects/*physiology, Quinoxalines/pharmacology, Rats, Receptors, Synapses/drug effects/physiology, Teyler T J
Gaussian Process Modeling of Protein Turnover.
Tags: *Brain Chemistry, *dynamic proteome, *Gaussian process, *Mass spectrometry, *Ornstein-Uhlenbeck process, *protein degradation rate constant, *protein turnover rate constant, *stable isotope labeling, *stochastic differential equation for protein turnover rate constant, 2016, Animals, Chromatography, Data Interpretation, Department of Pharmaceutical Sciences, Isotope Labeling, Journal of proteome research, Kasumov Takhar, Kinetics, Liquid, Liver/*chemistry, Mass spectrometry, Mice, NEOMED College of Pharmacy, Normal Distribution, Previs Stephen F, Proteins/*metabolism, Proteome/*metabolism, Proteomics/methods, Rahman Mahbubur, Sadygov Rovshan G, Statistical, Stochastic Processes
Expression and purification of human cholesterol 7 alpha-hydroxylase in Escherichia coli.
Tags: 1994, Animals, Base Sequence, Catalysis, Chiang J Y, Cholesterol 7-alpha-Hydroxylase/biosynthesis/genetics/*isolation & purification, Cytochrome P-450 Enzyme System/biosynthesis/isolation & purification, Department of Integrative Medical Sciences, Escherichia coli, Humans, Immunochemistry, Journal of lipid research, Karam W G, Kinetics, Molecular Sequence Data, NEOMED College of Medicine, Rats, Recombinant Proteins/biosynthesis, Solubility, Subcellular Fractions/enzymology
Estrogen differentially modulates nicotine-evoked dopamine release from the striatum of male and female rats.
Endogenous mGluR activity suppresses GABAergic transmission in avian cochlear nucleus magnocellularis neurons.
Tags: 2-Amino-5-phosphonovalerate/pharmacology, 2007, Amino Acids/pharmacology, Animals, Chickens/*physiology, Cochlear Nucleus/*cytology/*physiology, Department of Anatomy & Neurobiology, Electric Stimulation, Excitatory Amino Acid Antagonists/pharmacology, Excitatory Postsynaptic Potentials/physiology, GABA-B Receptor Agonists, GABA-B Receptor Antagonists, GABA-B/physiology, gamma-Aminobutyric Acid/*physiology, Glycine/analogs & derivatives/pharmacology, In Vitro Techniques, Journal of neurophysiology, Kinetics, Lu Yong, Membrane Potentials/drug effects, Metabotropic Glutamate/agonists/antagonists & inhibitors/*metabolism/physiology, Models, NEOMED College of Medicine, Neurological, Neurons/*physiology, Patch-Clamp Techniques, Receptors, Resorcinols/pharmacology, Synapses/physiology, Synaptic Transmission/*physiology, Xanthenes/pharmacology
Effects of cathinone and amphetamine on the neurochemistry of dopamine in vivo.
Tags: 1990, 3, 4-Dihydroxyphenylacetic Acid/metabolism, Alkaloids/*pharmacology, Amphetamine/*pharmacology, Animals, Brain/drug effects/*metabolism, Caudate Nucleus/metabolism, Dopamine/*metabolism, Homovanillic Acid/metabolism, Inbred Strains, Kinetics, Male, Molecular Structure, Neuropharmacology, Nucleus Accumbens/metabolism, Pehek E A, Psychotropic Drugs/*pharmacology, Putamen/metabolism, Rats, Reference Values, Schechter M D, Structure-Activity Relationship, Yamamoto B K
CONTINUOUS-INFUSION OF PYRIDOSTIGMINE IN THE MANAGEMENT OF MYASTHENIC CRISIS
Tags: 1993, Bonfiglio M F, cholinergic, cholinesterase inhibitors, compounds, Critical care medicine, edrophonium, General & Internal Medicine, gravis, Injections, Intravenous, Journal Article, Kinetics, Martin B R, myasthenia gravis, neostigmine, neuromuscular diseases, ocular motility disorders, pyridinium, pyridostigmine bromide, Receptors, Saltis L M, Traeger S M, ventilatory weaning
Castration reduces potassium-stimulated norepinephrine release from superfused olfactory bulbs of male rats.
Castration differentially alters [3H]nisoxetine binding to norepinephrine uptake sites in olfactory bulb and frontal cortex of male rats.
Tags: *Orchiectomy, 1999, Adrenergic/drug effects/*metabolism, Animals, Boja J W, Dluzen D E, Fluoxetine/*analogs & derivatives/metabolism, Frontal Lobe/drug effects/*metabolism, Kinetics, Male, Norepinephrine/metabolism, Olfactory Bulb/drug effects/*metabolism, Rats, Receptors, Shang Y, Sprague-Dawley, Synapse (New York, N.Y.), Synaptosomes/drug effects/metabolism, Testosterone/pharmacology
Analysis of the thymidine kinase of a herpes simplex virus type 1 isolate that exhibits resistance to (E)-5-(2-bromovinyl)-2'-deoxyuridine.
Tags: 1994, Acyclovir/pharmacology, Amino Acid Sequence, Antiviral Agents/metabolism/*pharmacology, Base Sequence, Binding Sites, Bromodeoxyuridine/*analogs & derivatives/metabolism/pharmacology, Deoxyuridine/analogs & derivatives/pharmacology, DNA, Docherty J J, Drug Resistance, Herpesvirus 1, Human/drug effects/*enzymology/genetics, Humans, Kinetics, Microbial, Molecular Sequence Data, Phosphonoacetic Acid/pharmacology, Phosphorylation, Point Mutation/genetics, Sequence Analysis, The Journal of general virology, Thymidine Kinase/genetics/metabolism, Thymidine/metabolism, Vidarabine/pharmacology, Wilber B A
A block in glycoprotein processing correlates with small plaque morphology and virion targetting to cell-cell junctions for an oral and an anal strain of herpes simplex virus type-1.
Tags: *Protein Processing, 1995, Anal Canal/virology, Animals, Archives of virology, Cercopithecus aethiops, Dick J W, Electron, Fluorescent Antibody Technique, Genetic Complementation Test, Herpesvirus 1, Human/genetics/isolation & purification/*physiology, Humans, Indirect, Intercellular Junctions/physiology/*virology, Kinetics, Microscopy, Mouth/virology, Post-Translational, Rosenthal K S, Species Specificity, Vero Cells, Viral Envelope Proteins/*biosynthesis/metabolism, Viral Plaque Assay, Virion/*physiology
3D-QSAR and docking studies of pentacycloundecylamines at the sigma-1 (sigma1) receptor.
Tags: *Quantitative Structure-Activity Relationship, 2013, Amines/*chemistry/metabolism, Aza Compounds/chemistry, Binding Sites, Bioorganic & medicinal chemistry letters, Geldenhuys Werner J, Kinetics, Malan Sarel F, Molecular Docking Simulation, Novotny Nicholas, Protein Binding, Protein Structure, Receptors, sigma/*chemistry/metabolism, Tertiary, Van der Schyf Cornelis J