Browse Items (132 total)
- Tags: Dose-Response Relationship
MDMA (Ecstasy) substitutes for the ethanol discriminative cue in HAD but not LAD rats.
Tags: 1995, 4-methylenedioxyamphetamine/*pharmacology, Alcohol (Fayetteville, N.Y.), Alcohol Drinking/*genetics/psychology, Animals, Central Nervous System Depressants/*pharmacology, Cues, Discrimination (Psychology)/*drug effects, Discrimination Learning/drug effects, Dose-Response Relationship, Drug, Ethanol/*pharmacology, Generalization, Gordon T L, Male, Meehan S M, N-Methyl-3, Piperazines/pharmacology, Rats, Schechter M D, Serotonin Agents/*pharmacology, Serotonin Receptor Agonists/pharmacology, Stimulus
Resveratrol inhibition of varicella-zoster virus replication in vitro.
Tags: 2006, Antiviral Agents/*pharmacology, Antiviral research, Bailey Erin, Blotting, Booth Tristan, Cell Line, Docherty John J, Dose-Response Relationship, Drug, Faith Seth A, Fibroblasts/virology, Herpesvirus 3, Human/*drug effects/physiology, Humans, Immediate-Early Proteins/biosynthesis, Messenger/biosynthesis, Resveratrol, Reverse Transcriptase Polymerase Chain Reaction, RNA, Stilbenes/*pharmacology, Sweet Thomas J, Trans-Activators/biosynthesis, Viral Envelope Proteins/biosynthesis, Viral Plaque Assay, Viral/biosynthesis, Virus Attachment/drug effects, Virus Inactivation/drug effects, Virus Replication/*drug effects, Western
A standardized extract of Butea monosperma (Lam.) flowers suppresses the
Tags: *Butea, 2017, Aged, Ansari Mohammad Y, Autophagy, Autophagy/drug effects/physiology, Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, Butea monosperma (Lam.), Chondrocytes/drug effects/*metabolism, Department of Anatomy & Neurobiology, Dose-Response Relationship, Drug, Flowers, Gene Expression, Haqqi Tariq M, Humans, Interleukin-1beta/*pharmacology, Interleukin-6/*biosynthesis/genetics, Khan Nazir M, Matrix Metalloproteinase 13/biosynthesis/genetics, Matrix Metalloproteinase 3/biosynthesis/genetics, Matrix Metalloproteinase 9/biosynthesis/genetics, Matrix Metalloproteinases/*biosynthesis/genetics, Middle Aged, mTOR, NEOMED College of Medicine, Nutraceuticals, Osteoarthritis, Osteoarthritis/*metabolism, Plant Extracts/isolation & purification/pharmacology
Structure-based design of a thiazolidinedione which targets the mitochondrial protein mitoNEET.
Tags: *Drug Design, 2010, Animals, Barnes Kendra F, Binding Sites/drug effects/physiology, Bioorganic & medicinal chemistry letters, Carroll Richard T, Dose-Response Relationship, Drug, Drug Delivery Systems/*methods, Funk Max O, Geldenhuys Werner J, Liver/drug effects/metabolism, Mitochondria, Mitochondrial Proteins/*metabolism, Protein Structure, Rats, Secondary, Structure-Activity Relationship, Thiazolidinediones/administration & dosage/*chemical synthesis/*metabolism
A novel binding assay identifies high affinity ligands to the rosiglitazone binding site of mitoNEET.
Tags: 2011, Awale Prabha S, Binding Sites/drug effects, Bioorganic & medicinal chemistry letters, Carroll Richard T, Dose-Response Relationship, Drug, Funk Max O, Geldenhuys Werner J, Ligands, Lin Li, Mitochondrial Proteins/*antagonists & inhibitors/metabolism, Molecular Structure, Recombinant Proteins/antagonists & inhibitors/metabolism, Rosiglitazone, Stereoisomerism, Structure-Activity Relationship, Thiazolidinediones/chemical synthesis/chemistry/*pharmacology
Screening and identification of novel compounds with potential anti-proliferative effects on gallium-resistant lung cancer through an AXL kinase pathway.
Tags: 2014, Alazizi Adnan, Antineoplastic Agents/chemical synthesis/chemistry/*pharmacology, Antitumor, AXL, Bioorganic & medicinal chemistry letters, Cell Line, Cell Proliferation/drug effects, Cell Survival/drug effects, Department of Pharmaceutical Sciences, Dose-Response Relationship, Drug, Drug Resistance, Drug Screening Assays, Gallium, Gallium-resistance, Gallium/pharmacology, Geldenhuys Werner J, Humans, Lin Li, Liva Sophia, Lung cancer, Lung Neoplasms/drug therapy/*enzymology/*pathology, Molecular Structure, Naphthalenes/chemistry/*pharmacology, NEOMED College of Pharmacy, Neoplasm/drug effects, Oyewumi Moses O, Proto-Oncogene Proteins/*antagonists & inhibitors/metabolism, Pyrazoles/chemistry/*pharmacology, Quinolines/chemistry/*pharmacology, Receptor Protein-Tyrosine Kinases/*antagonists & inhibitors/metabolism, Structure-Activity Relationship, Tetrazoles/chemistry/*pharmacology, Tumor, Virtual screening
Structure-activity and in vivo evaluation of a novel lipoprotein lipase (LPL) activator.
Tags: *Diabetes, *High-fat diet, *Homology modeling, *Hyperlipidemia, *Lipoprotein lipase, *Liver cirrhosis, *Obesity, 2017, Animals, Benzeneacetamides/chemical synthesis/chemistry/*pharmacology, Bioorganic & medicinal chemistry letters, Caporoso Joel, Darvesh Altaf S, Department of Integrative Medical Sciences, Department of Pharmaceutical Sciences, Department of Pharmacy Practice, Dose-Response Relationship, Drug, Geldenhuys Werner J, Imidazoles/chemical synthesis/chemistry/*pharmacology, Lee Yoon-Kwang, Leeper Thomas C, Lin Li, Lipoprotein Lipase/*metabolism, Mice, Molecular Docking Simulation, Molecular Structure, NEOMED College of Graduate Studies, NEOMED College of Medicine, NEOMED College of Pharmacy, Sadana Prabodh, Structure-Activity Relationship
Resveratrol-mediated chemoprevention of diethylnitrosamine-initiated hepatocarcinogenesis: inhibition of cell proliferation and induction of apoptosis.
Tags: 2009, Animal, Animals, Anticarcinogenic Agents/*antagonists & inhibitors/pharmacology, Antitumor, Apoptosis/*drug effects, Bishayee Anupam, Body Weight/drug effects, Cell Proliferation/drug effects, Chemico-biological interactions, Dhir Neetika, Diethylnitrosamine, Disease Models, Dose-Response Relationship, Drinking/drug effects, Drug, Drug Screening Assays, Eating/drug effects, Experimental/chemically induced/pathology/*prevention & control, Female, Immunohistochemistry, Liver Neoplasms, Organ Size/drug effects, Phenobarbital, Proto-Oncogene Proteins c-bcl-2/biosynthesis, Rats, Resveratrol, Sprague-Dawley, Stilbenes/*pharmacology
Formulation and photoirradiation parameters that influenced photoresponsive drug delivery using alkoxylphenacyl-based polycarbonates.
Tags: 2014, Animals, Biocompatibility, Cardiotoxicity, Cell Line, Chamsaz Elaheh A, Chemistry, Department of Pharmaceutical Sciences, Dose-Response Relationship, Doxorubicin, Drug, Drug Delivery Systems/*methods, European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V, Heart/drug effects, Humans, Inbred BALB C, Joy Abraham, Mice, Nanotechnology, NEOMED College of Pharmacy, Oyewumi Moses O, Pharmaceutical, Photic Stimulation/*methods, Photoresponsive, Photosensitizing Agents/*chemical synthesis/radiation effects/toxicity, Polycarboxylate Cement/*chemical synthesis/radiation effects/toxicity, Polymer chain scission, Stimuli-responsive, Tumor, Wehrung Daniel
The role of the N-terminal and mid-region residues of substance P in regulating functional selectivity at the tachykinin NK1 receptor.
Tags: 2008, Amino Acid Sequence, Animals, Beard Debbie J, Binding, Calcium Signaling/physiology, CHO Cells, Competitive/drug effects, Cricetinae, Cricetulus, Dose-Response Relationship, Drug, European journal of pharmacology, Iodine Radioisotopes, Ligands, Models, Molecular, Molecular Sequence Data, Neurokinin-1/chemistry/drug effects/*metabolism, Perrine Shane A, Rats, Receptors, Simmons Mark A, Substance P/chemistry/drug effects/*physiology, Young John K
The effect of gender and the neurotrophin, BDNF, upon methamphetamine-induced neurotoxicity of the nigrostriatal dopaminergic system in mice.
Tags: 2004, Animals, Brain-Derived Neurotrophic Factor/deficiency/genetics/*metabolism, Central Nervous System Stimulants/poisoning, Corpus Striatum/*drug effects/*metabolism, Dluzen Dean E, Dopamine/*metabolism, Dose-Response Relationship, Drug, Female, Humans, Male, Methamphetamine/*poisoning, Mice, Mutation, Neuroscience letters, Neurotoxicity Syndromes/*etiology/*metabolism, Sex Factors, Structure-Activity Relationship, Substantia Nigra/drug effects/metabolism, Transgenic
Testosterone enhances dopamine depletion by methamphetamine in male, but not female, mice.
Tags: *Sex Characteristics, 2008, Animals, Castration/methods, Corpus Striatum/drug effects/metabolism, Dluzen Dean E, Dopamine Uptake Inhibitors/*pharmacology, Dopamine/*metabolism, Dose-Response Relationship, Drug, Female, Lewis Chandani, Male, Methamphetamine/*pharmacology, Mice, Neuroscience letters, Testosterone Propionate/*pharmacology
Valproate increases dopamine transporter expression through histone acetylation and enhanced promoter binding of Nurr1.
Tags: 2017, Acetylation/drug effects, Animals, Butyrates/pharmacology, Cell Line, Cell Survival/drug effects, Department of Pharmaceutical Sciences, Dopamine Plasma Membrane Transport Proteins/*metabolism, Dopamine transporter, Dopaminergic Neurons/cytology/drug effects/metabolism, Dose-Response Relationship, Drug, Eid Aseel, Epigenesis, Epigenetics, Genetic, Genetic/drug effects, Green Ashley L, Group A, Guo Grace L, HDAC, Histone deacetylase, Histone Deacetylase Inhibitors/*pharmacology, Histone Deacetylases/metabolism, Histones/*drug effects/metabolism, Homeodomain Proteins/metabolism, Hydroxamic Acids/pharmacology, Member 2/*metabolism, Messenger/metabolism, NEOMED College of Pharmacy, Neuropharmacology, Nuclear Receptor Subfamily 4, Nurr1, Pitx3, Promoter Regions, Rats, Richardson Jason R, RNA, Transcription Factors/metabolism, Valproate, Valproic Acid/*pharmacology, Zarbl Helmut, Zhan Le
Localization and function of NK(3) subtype tachykinin receptors of layer V pyramidal neurons of the guinea-pig medial prefrontal cortex.
Tags: 2008, Animals, Autoradiography/methods, Dose-Response Relationship, Drug, Drug Interactions, Excitatory Amino Acid Antagonists/pharmacology, Excitatory Postsynaptic Potentials/drug effects/radiation effects, Guinea Pigs, In Vitro Techniques, Iodine Isotopes/pharmacokinetics, Male, Medd A M, Membrane Potentials/drug effects/physiology/radiation effects, Neurokinin B/analogs & derivatives/pharmacokinetics, Neurokinin-3/agonists/antagonists & inhibitors/*metabolism, Neuroscience, Patch-Clamp Techniques, Peptide Fragments/pharmacology, Prefrontal Cortex/*cytology, Protein Binding/drug effects, Pyramidal Cells/drug effects/*metabolism, Quinolines/pharmacology, Quinoxalines/pharmacology, Receptors, Simmons M A, Sobotka-Briner C D, Substance P/analogs & derivatives/pharmacology, Valine/analogs & derivatives/pharmacology
A subtherapeutic international normalized ratio despite increasing doses of warfarin: could this be malabsorption?
Tags: *Drug Resistance, 2000, Administration, Adult, Anticoagulants/administration & dosage/metabolism/pharmacokinetics/therapeutic use, Area Under Curve, Biological Availability, Delgado L L, Department of Family & Community Medicine, Department of Internal Medicine, Dose-Response Relationship, Drug, Female, Frazee L A, Haupt K M, Humans, Injections, Intestinal Absorption/*physiology, Intravenous, Kidney Transplantation, Lara L F, NEOMED College of Medicine, Oral, Rutecki G W, The American journal of the medical sciences, Warfarin/*administration & dosage/*metabolism/pharmacokinetics/therapeutic use
Discrimination of cocaethylene in rats trained to discriminate between its components.
Olanzapine attenuates the reinforcing effects of cocaine.
Tags: 1997, Animal/*drug effects, Animals, Antipsychotic Agents/administration & dosage/*pharmacology, Behavior, Benzodiazepines, Cocaine/administration & dosage/antagonists & inhibitors/*pharmacology, Conditioning, Dopamine Uptake Inhibitors/administration & dosage/*pharmacology, Dose-Response Relationship, Drug, European journal of pharmacology, Food Preferences/drug effects, Male, Meil W M, Olanzapine, Operant/*drug effects, Pirenzepine/administration & dosage/*analogs & derivatives/pharmacology, Rats, Schechter M D, Self Administration, Sprague-Dawley
The effects of nicotine on dopamine and DOPAC output from rat striatal tissue.
Tags: 1998, 3, 4-Dihydroxyphenylacetic Acid/*metabolism, Amphetamine/pharmacology, Anderson L I, Animals, Central Nervous System Stimulants/pharmacology, Corpus Striatum/*drug effects/*metabolism, Dluzen D E, Dopamine/*metabolism, Dose-Response Relationship, Drug, European journal of pharmacology, Ganglionic Stimulants/administration & dosage/*pharmacology, Male, Nicotine/administration & dosage/*pharmacology, Potassium Chloride/pharmacology, Rats, Sprague-Dawley
Discrete versus cumulative dosing in dose-response discrimination studies.
Tags: 1997, 4-methylenedioxyamphetamine/*pharmacology, Animals, Chemical, Cocaine/*pharmacology, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Drug Administration Schedule, Drug Evaluation, European journal of pharmacology, Male, N-Methyl-3, Preclinical, Rats, Schechter M D, Sprague-Dawley, Stimulation
Sex differences in extracellular and intracellular calcium-mediated vascular reactivity to vasopressin in rat aorta.
Tags: *Sex Characteristics, 1, 1998, 3-Pyridinecarboxylic acid, 4-dihydro-2, 6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Animals, Aorta/drug effects/*metabolism, Calcium Channel Agonists/*pharmacology, Calcium Channel Blockers/*pharmacology, Calcium/*metabolism, Department of Internal Medicine, Diltiazem/pharmacology, Dose-Response Relationship, Drug, Eatman D, European journal of pharmacology, Female, In Vitro Techniques, Male, Methyl ester/pharmacology, NEOMED College of Medicine, Potassium Chloride/pharmacology, Rats, Rutecki G W, Simvastatin/pharmacology, Sprague-Dawley, Stallone J N, Vasoconstriction/*drug effects, Vasopressins/*metabolism, Whittier F C
Phentermine+fenfluramine produce cocaine-like discriminative cues.
Tags: *Discrimination (Psychology), 1996, Animals, Cocaine/*pharmacology, Department of Anatomy & Neurobiology, Dose-Response Relationship, Drug, Fenfluramine/administration & dosage/*pharmacology, Life sciences, Male, McBurney D, NEOMED College of Medicine, Phentermine/administration & dosage/*pharmacology, Rats, Schechter M D, Sprague-Dawley
Serotonergic mediation of fenfluramine discriminative stimuli in fawn-hooded rats.
Tags: *Discrimination Learning, 1997, 4-methylenedioxyamphetamine/pharmacology, Animals, Dose-Response Relationship, Drug, Fenfluramine/administration & dosage/*pharmacology, Fluoxetine/pharmacology, Ibogaine/pharmacology, Life sciences, Male, Methoxydimethyltryptamines/pharmacology, N-Methyl-3, Piperazines/pharmacology, Quipazine/pharmacology, Rats, Schechter M D, Serotonin Agents/administration & dosage/*pharmacology, Serotonin Receptor Agonists/pharmacology, Serotonin/*metabolism, Sprague-Dawley
Drug-drug discrimination: stimulus properties of drugs of abuse upon a serotonergic-dopaminergic continuum.
Tags: 1997, 4-methylenedioxyamphetamine/pharmacology, Amphetamine/pharmacology, Animals, Discrimination (Psychology)/*drug effects, Dopamine Agonists/pharmacology, Dopamine Uptake Inhibitors/pharmacology, Dopamine/*physiology, Dose-Response Relationship, Drug, Generalization, Lysergic Acid Diethylamide/pharmacology, Male, N-Methyl-3, Norfenfluramine/pharmacology, Pharmacology, biochemistry, and behavior, Propiophenones/pharmacology, Rats, Schechter M D, Serotonin Agents/pharmacology, Serotonin Receptor Agonists/pharmacology, Serotonin Uptake Inhibitors/pharmacology, Serotonin/*physiology, Stimulus, Substance-Related Disorders/*psychology, Tetrahydronaphthalenes/pharmacology, Time Factors
Discriminative characteristics of high and low cocaine administration: effect of other psychostimulants.
Tags: 1997, Amphetamine/pharmacology, Animals, Central Nervous System Stimulants/pharmacology, Cocaine/*pharmacology, Conditioning, Discrimination Learning/*drug effects, Dopamine Agents/*pharmacology, Dose-Response Relationship, Drug, Drug Evaluation, Generalization, Male, Methamphetamine/pharmacology, Operant/*drug effects, Pharmacology, biochemistry, and behavior, Preclinical, Propiophenones/pharmacology, Psychotropic Drugs/*pharmacology, Rats, Response/*drug effects, Schechter M D
Rohypnol ("roofies") control of drug discrimination: effect of coadministered ethanol or flumenazil.
Tags: 1998, Animals, Anti-Anxiety Agents/*pharmacology, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Drug Administration Schedule, Ethanol/*pharmacology, Flumazenil/*pharmacology, Flunitrazepam/*pharmacology, GABA Antagonists/*pharmacology, Male, Pharmacology, biochemistry, and behavior, Rats, Schechter M D, Sprague-Dawley
MDMA-like stimulus effects of hallucinogens in male Fawn-Hooded rats.
Tags: 1998, 4-methylenedioxyamphetamine/*pharmacology, Animals, Central Nervous System Stimulants/*pharmacology, Conditioning, Cues, Discrimination (Psychology)/drug effects, Dopamine Agents/pharmacology, Dose-Response Relationship, Drug, Generalization, Hallucinogens/*pharmacology, Inbred Strains, Male, N-Methyl-3, Operant/drug effects, Pharmacology, biochemistry, and behavior, Rats, Schechter M D, Serotonin Agents/pharmacology, Serotonin/genetics/physiology, Sprague-Dawley, Stimulus/drug effects
Secure cranial-mount intrathecal cannulation - a spinal administration technique in the rat.
Tags: 2000, Analgesics, Anesthesia, Animals, Crisp T, Dose-Response Relationship, Drug, Injections, Journal of neuroscience methods, Microinjections, Morphine/administration & dosage/pharmacology, Opioid/administration & dosage/pharmacology, Rats, Schechter J B, Spinal Cord/*physiology, Spinal/*instrumentation, Sprague-Dawley, Stereotaxic Techniques/*instrumentation
Resveratrol inhibition of Propionibacterium acnes.
Tags: *Anti-Bacterial Agents, 2007, Anti-Inflammatory Agents, Bailey Erin, Benzoyl Peroxide/pharmacology, Booth Tristan D, Department of Family & Community Medicine, Docherty John J, Dose-Response Relationship, Drug, Erythromycin/pharmacology, Keratolytic Agents/pharmacology, McEwen Heather A, Microbial Sensitivity Tests, NEOMED College of Medicine, Non-Steroidal/*pharmacology, Propionibacterium acnes/*drug effects/growth & development, Resveratrol, Stilbenes/*pharmacology, Sweet Thomas J, The Journal of antimicrobial chemotherapy
Selective Targeting of Heme Protein in Cytochrome P450 and Nitric Oxide Synthase by Diphenyleneiodonium.
Tags: *cytochrome P450, *flavoenzymes, *heme, *nitric oxide synthase, *Reactive oxygen species, 2016, Aleksunes Lauren M, Animals, Cytochrome P-450 Enzyme Inhibitors/*pharmacology, Cytochrome P-450 Enzyme System/*metabolism, Department of Pharmaceutical Sciences, Dose-Response Relationship, Drug, Heck Diane E, Heindel Ned D, Heme/*antagonists & inhibitors/metabolism, Humans, Jan Yi-Hua, Laskin Debra L, Laskin Jeffrey D, Liver/drug effects/enzymology, Mice, Microsomes, Mishin Vladimir, NEOMED College of Pharmacy, Nitric Oxide Synthase Type II/*antagonists & inhibitors/metabolism, Nitric Oxide/metabolism, Onium Compounds/*pharmacology, Rats, Recombinant Proteins/metabolism, Richardson Jason R, Sprague-Dawley, Szilagyi John T, Time Factors, Toxicological sciences : an official journal of the Society of Toxicology
Pyrethroid Insecticides Directly Activate Microglia Through Interaction With Voltage-Gated Sodium Channels.
Tags: *deltamethrin, *intracellular sodium., *Microglia, *neurodegeneration, *Neuroinflammation, *permethrin, *pyrethroids, *tetrodotoxin, *tumor necrosis factor, *Voltage-gated sodium channels, 2017, Animals, Cell Line, Department of Pharmaceutical Sciences, Dose-Response Relationship, Drug, Hossain Muhammad M, Inbred C57BL, Insecticides/*toxicity, Ion Channel Gating/*drug effects, Liu Jason, Mice, Microglia/*drug effects/metabolism, NEOMED College of Pharmacy, Pyrethrins/*toxicity, Richardson Jason R, Sodium Channels/*drug effects, Toxicological sciences : an official journal of the Society of Toxicology, Transformed, Tumor Necrosis Factor-alpha/metabolism
Evaluation of factors associated with achieving glycemic control in a pharmacist-managed diabetes clinic.
Tags: 2014, Ambulatory Care, Ambulatory Care/organization & administration, American journal of therapeutics, Blood Glucose – Drug Effects, Blood Glucose/drug effects, Boros Melanie L, Department of Internal Medicine, Department of Pharmaceutical Sciences, Department of Pharmacy Practice, Diabetes Mellitus, Dose-Response Relationship, Drug, Female, Follow-Up Studies, Frazee Lawrence A, Glycated Hemoglobin A/metabolism, Glycosylated – Metabolism, Hemoglobin A, Human, Humans, Hypoglycemic Agents – Administration and Dosage, Hypoglycemic Agents – Therapeutic Use, Hypoglycemic Agents/administration & dosage/*therapeutic use, Insulin – Administration and Dosage, Insulin – Therapeutic Use, Insulin/administration & dosage/therapeutic use, Kostoff Matthew D, Male, Middle Age, Middle Aged, Moorman John M, NEOMED College of Medicine, NEOMED College of Pharmacy, Pharmaceutical Services/*organization & administration, Pharmacists – Administration, Pharmacists/*organization & administration, Pharmacy Service – Administration, Prospective Studies, Retrospective Design, Retrospective Studies, Social Work – Statistics and Numerical Data, Social Work/statistics & numerical data, Treatment Outcome, Treatment Outcomes, Type 2 – Drug Therapy, Type 2/*drug therapy
Activation of metabotropic glutamate receptor 1 dimers requires glutamate binding in both subunits.
Tags: 2005, Blotting, Calcium Channels/drug effects/metabolism, Department of Integrative Medical Sciences, DNA/biosynthesis/genetics, Dose-Response Relationship, Drug, Fluorescent Antibody Technique, Genes, Glutamic Acid/*metabolism, Humans, Kammermeier Paul J, Membrane Potentials/drug effects, Metabotropic Glutamate/genetics/*metabolism, myc/genetics, NEOMED College of Medicine, Patch-Clamp Techniques, Plasmids/genetics, Receptors, Signal Transduction/drug effects, Superior Cervical Ganglion/cytology/drug effects/metabolism, Sympathetic Nervous System/cytology/drug effects/metabolism, The Journal of pharmacology and experimental therapeutics, Western, Yun June
Functional selectivity of NK1 receptor signaling: peptide agonists can preferentially produce receptor activation or desensitization.
Tags: 2006, Animals, CHO Cells, Cricetinae, Dose-Response Relationship, Drug, Humans, Neurokinin-1/agonists/drug effects/*physiology, Rana catesbeiana, Rats, Receptors, Signal Transduction/*physiology, Simmons Mark A, Substance P/metabolism/pharmacology, Tachykinins/metabolism/pharmacology, The Journal of pharmacology and experimental therapeutics
Endothelin-mediated in vivo pressor responses following TRPV1 activation.
Tags: *Blood Pressure/drug effects, *Vasoconstriction/drug effects, 2011, Adrenergic alpha-Agonists/administration & dosage, American journal of physiology. Heart and circulatory physiology, Analysis of Variance, Animal, Animals, Azepines/administration & dosage, Biphenyl Compounds/administration & dosage, Bratz Ian N, Capsaicin/administration & dosage, Cells, Cultured, Damron Derek S, Department of Integrative Medical Sciences, Diabetes Mellitus, Diabetic Angiopathies/genetics/*metabolism/physiopathology, Dipeptides/administration & dosage, Disease Models, Dose-Response Relationship, Drug, Endothelial Cells/metabolism, Endothelin A Receptor Antagonists, Endothelin A/metabolism, Endothelin B Receptor Antagonists, Endothelin B/metabolism, Endothelin-1/*metabolism, Enzyme-Linked Immunosorbent Assay, Femoral Artery/drug effects/*metabolism/physiopathology, Guarini Giacinta, Haney Rebecca M, Inbred C57BL, Indoles/administration & dosage, Infusions, Intravenous, Knockout, Male, Meszaros J Gary, Mice, NEOMED College of Medicine, Ohanyan Vahagn A, Phenylephrine/administration & dosage, Raman Priya, Receptor, Talasila Phani K, Thodeti Charles K, TRPV Cation Channels/agonists/deficiency/genetics/*metabolism, Type 2/genetics/*metabolism/physiopathology, Vasoconstrictor Agents/administration & dosage
Sexual dimorphism in vasopressin-induced contraction of rat aorta.
Acute exercise enhances nitric oxide modulation of vascular response to phenylephrine.
Tags: *Physical Exertion, 1993, Animals, Arginine/analogs & derivatives/pharmacology, Blood Flow Velocity, Blood Pressure/drug effects, Blood Vessels/*drug effects, Collins H L, DiCarlo S E, Dose-Response Relationship, Drug, Female, Heart Rate/drug effects, Iliac Artery/drug effects/physiology, Male, NG-Nitroarginine Methyl Ester, Nitric Oxide/antagonists & inhibitors/*physiology, Patil R D, Phenylephrine/*pharmacology, Rats, Sprague-Dawley, The American journal of physiology, Time Factors, Vasoconstriction/drug effects/physiology
Myocardial work load is a major determinant of norepinephrine-induced left ventricular dysfunction.
Tags: 1994, Allman F D, Anesthesia, Animals, Blood Pressure/*drug effects, Bosso F J, Cardiovascular, Consciousness, Diastole/drug effects, Dose-Response Relationship, Drug, General, Heart Rate/*drug effects, Heart/drug effects/*physiology, Left/drug effects/*physiology, Models, Norepinephrine/*pharmacology, Pentobarbital, Pilati C F, Rabbits, Systole/drug effects, The American journal of physiology, Time Factors, Ventricular Function
RNA interference for alpha-ENaC inhibits rat lung fluid absorption in vivo.
Tags: 2006, Absorption/drug effects, Adrenergic beta-Agonists/pharmacology, American journal of physiology. Lung cellular and molecular physiology, Amiloride/pharmacology, Animals, Body Fluids/*metabolism, Capillary Permeability, Dose-Response Relationship, Drug, Endothelium, Epithelial Cells/metabolism, Epithelial Sodium Channels, Epithelium/metabolism, Folkesson Hans G, Inhibitory Concentration 50, Li Tianbo, Lung/enzymology/*metabolism, Male, Messenger/antagonists & inhibitors/metabolism, Permeability, Plasmids/administration & dosage/pharmacology, Rats, RNA, Small Interfering/genetics/pharmacology, Sodium Channels/drug effects/genetics/metabolism/*physiology, Sprague-Dawley, Terbutaline/pharmacology, Tissue Distribution, Vascular/metabolism
Mesenteric vascular responses to vasopressin during development of DOCA-salt hypertension in male and female rats.
Tags: 1995, 6-Ketoprostaglandin F1 alpha/metabolism, Analysis of Variance, Animals, Arginine Vasopressin/*pharmacology, Blood Pressure/drug effects, Desoxycorticosterone, Dietary, Dinoprostone/metabolism, Dose-Response Relationship, Drug, Female, Hypertension/chemically induced/*physiopathology, In Vitro Techniques, Male, Prostaglandins/analysis/*metabolism, Rats, Reference Values, Sex Characteristics, Sodium, Splanchnic Circulation/drug effects/*physiology, Sprague-Dawley, Stallone J N, The American journal of physiology
Reduced vascular responsiveness after a single bout of dynamic exercise in the conscious rabbit.
Tags: 1992, Adenosine/pharmacology, Adrenergic/physiology, Animals, Blood Vessels/*physiology, DiCarlo S E, Dose-Response Relationship, Drug, Hindlimb/physiology, Howard M G, In Vitro Techniques, Isoproterenol/pharmacology, Journal of applied physiology (Bethesda, Md. : 1985), Phenylephrine/pharmacology, Physical Exertion/*physiology, Pressoreceptors/physiology, Purinergic/physiology, Rabbits, Receptors, Reflex/physiology, Regional Blood Flow/physiology