Browse Items (129 total)
- Tags: Drug
Acute exercise attenuates phenylephrine-induced contraction of rabbit isolated aortic rings.
Tags: *Physical Conditioning, 1992, Adrenergic, alpha/physiology, Animal, Animals, Aorta/physiology, DiCarlo S E, Dose-Response Relationship, Drug, Howard M G, In Vitro Techniques, Medicine and science in sports and exercise, Muscle, Muscle Contraction/*drug effects, Phenylephrine/*pharmacology, Rabbits, Receptors, Smooth, Stallone J N, Vascular/*drug effects/physiology
Preferential increase in pituitary prolactin versus vasoactive intestinal peptide as a function of estradiol benzoate dose in the ovariectomized rat.
Tags: 1991, Animals, Brain/drug effects/*metabolism, Carrillo A J, Doherty P C, Dose-Response Relationship, Drug, Endocrinology, Estradiol/*pharmacology, Female, Guan X B, Inbred Strains, Organ Specificity, Ovariectomy, Pituitary Gland/drug effects/*metabolism, Prolactin/blood/*metabolism, Rats, Sturtevant J R, Thyrotropin/blood/metabolism, Vasoactive Intestinal Peptide/*metabolism, Walro D G
Antitumor efficacy and tolerability of systemically administered gallium acetylacetonate-loaded gelucire-stabilized nanoparticles.
Tags: *Lethal Dose 50, 2013, Adenocarcinoma/*drug therapy/pathology, Animals, Antineoplastic Agents/administration & dosage/pharmacokinetics/toxicity, Bi Lipeng, Cell Line, Department of Pharmaceutical Sciences, Dose-Response Relationship, Drug, Drug Stability, Drug Tolerance, Gallium/*administration & dosage/pharmacokinetics/*toxicity, Geldenhuys Werner J, Humans, Journal of biomedical nanotechnology, Metabolic Clearance Rate, Mice, Nanocapsules/*administration & dosage/chemistry/*toxicity, NEOMED College of Pharmacy, Nude, Organ Specificity, Oyewumi Moses O, Tissue Distribution, Treatment Outcome, Triglycerides/chemistry, Tumor, Wehrung Daniel
An open-label dose escalation study to evaluate the safety of administration of nonviral stromal cell-derived factor-1 plasmid to treat symptomatic ischemic heart failure.
Tags: *Plasmids, 2013, Aged, Aras Rahul, Brain/blood, Chemokine CXCL12/*genetics/metabolism, Circulation research, Clemens Ruth, Cohort Studies, Dose-Response Relationship, Drug, Echocardiography, Exercise Tolerance, Farr Maryjane, Female, Follow-Up Studies, Genetic Therapy/*adverse effects/*methods, Heart Failure/metabolism/pathology/*therapy, Humans, Losordo Douglas W, Male, Mendelsohn Farrell O, Middle Aged, Myocardium/metabolism/pathology, Natriuretic Peptide, Pastore Joseph, Penn Marc S, Peptide Fragments/blood, Positron-Emission Tomography, Quality of Life, Rouy Didier, Schaer Gary L, Sherman Warren, Treatment Outcome
Effects of estrogen and related agents upon methamphetamine-induced neurotoxicity within an impaired nigrostriatal dopaminergic system of ovariectomized mice.
Tags: 2006, 3, 4-Dihydroxyphenylacetic Acid/metabolism, Androgens/administration & dosage, Animals, Dluzen Dean E, Dopamine Agents/*administration & dosage/toxicity, Dopamine/metabolism, Dose-Response Relationship, Drug, Drug Administration Schedule, Estradiol/administration & dosage/*analogs & derivatives/physiology, Estrogen Antagonists/administration & dosage, Female, Liu Bin, Methamphetamine/*administration & dosage/toxicity, Mice, Neostriatum/*drug effects/metabolism, Nerve Degeneration/chemically induced/prevention & control, Neuroendocrinology, Neuroprotective Agents/administration & dosage, Neurotoxins/*administration & dosage, Ovariectomy, Parkinson Disease/physiopathology, Substantia Nigra/*drug effects/metabolism, Tamoxifen/administration & dosage
Dose-response effects of estrogen and tamoxifen upon methamphetamine-induced behavioral responses and neurotoxicity of the nigrostriatal dopaminergic system in female mice.
Tags: 2004, 3, 4-Dihydroxyphenylacetic Acid/metabolism, Animal/*drug effects, Animals, Behavior, Brain Chemistry/drug effects, Dluzen Dean E, Dopamine/*metabolism, Dose-Response Relationship, Drug, Drug Interactions, Estrogen Antagonists/pharmacology, Estrogens/*pharmacology, Female, Methamphetamine/*toxicity, Mice, Mickley Katherine R, Movement/drug effects, Neostriatum/*drug effects/physiology, Neuroendocrinology, Neurotoxins/*toxicity, Organ Size/drug effects, Ovariectomy/methods, Stereotyped Behavior/drug effects, Substantia Nigra/drug effects/physiology, Tamoxifen/*pharmacology, Uterus
Resveratrol suppresses oxidative stress and inflammatory response in diethylnitrosamine-initiated rat hepatocarcinogenesis.
Tags: 2010, Animals, Antioxidants/*pharmacology/therapeutic use, Antitumor, Barnes Kendra F, Bhatia Deepak, Bishayee Anupam, Cancer prevention research (Philadelphia, Pa.), Carcinogens/toxicity, Carroll Richard T, Chemical and Drug Induced Liver Injury/*etiology/metabolism/pathology, Darvesh Altaf S, Department of Pharmaceutical Sciences, Diethylnitrosamine/toxicity, Dose-Response Relationship, Drug, Drug Screening Assays, Enzyme Induction/drug effects, Experimental/chemically induced/metabolism/pathology/*prevention & control, Female, Hyperplasia, Inflammation/*prevention & control, Lipid Peroxidation/drug effects, Liver Neoplasms, Liver/drug effects/metabolism/pathology, Messenger/biosynthesis/genetics, NEOMED College of Pharmacy, NF-E2-Related Factor 2/biosynthesis/genetics, Nitric Oxide Synthase Type II/biosynthesis/genetics, Oxidative Stress/*drug effects, Phenobarbital/toxicity, Precancerous Conditions/*chemically induced/metabolism/pathology, Rats, Resveratrol, RNA, Sprague-Dawley, Stilbenes/*pharmacology/therapeutic use, Tyrosine/analogs & derivatives/analysis
Dose-response relationship between plasma epinephrine concentration and alveolar liquid clearance in dogs.
Tags: 1998, Algorithms, Animals, Blood Pressure/drug effects/physiology, Cardiac Output/drug effects/physiology, Catecholamines/blood, Dogs, Dose-Response Relationship, Drug, Epinephrine/*blood, Female, Hematocrit, Journal of applied physiology (Bethesda, Md. : 1985), Male, Maron M B, Pulmonary Alveoli/*physiopathology, Pulmonary Circulation/drug effects/physiology, Pulmonary Edema/*blood/*physiopathology, Pulmonary Wedge Pressure/drug effects/physiology
Reduced vascular responsiveness after a single bout of dynamic exercise in the conscious rabbit.
Tags: 1992, Adenosine/pharmacology, Adrenergic/physiology, Animals, Blood Vessels/*physiology, DiCarlo S E, Dose-Response Relationship, Drug, Hindlimb/physiology, Howard M G, In Vitro Techniques, Isoproterenol/pharmacology, Journal of applied physiology (Bethesda, Md. : 1985), Phenylephrine/pharmacology, Physical Exertion/*physiology, Pressoreceptors/physiology, Purinergic/physiology, Rabbits, Receptors, Reflex/physiology, Regional Blood Flow/physiology
Mesenteric vascular responses to vasopressin during development of DOCA-salt hypertension in male and female rats.
Tags: 1995, 6-Ketoprostaglandin F1 alpha/metabolism, Analysis of Variance, Animals, Arginine Vasopressin/*pharmacology, Blood Pressure/drug effects, Desoxycorticosterone, Dietary, Dinoprostone/metabolism, Dose-Response Relationship, Drug, Female, Hypertension/chemically induced/*physiopathology, In Vitro Techniques, Male, Prostaglandins/analysis/*metabolism, Rats, Reference Values, Sex Characteristics, Sodium, Splanchnic Circulation/drug effects/*physiology, Sprague-Dawley, Stallone J N, The American journal of physiology
RNA interference for alpha-ENaC inhibits rat lung fluid absorption in vivo.
Tags: 2006, Absorption/drug effects, Adrenergic beta-Agonists/pharmacology, American journal of physiology. Lung cellular and molecular physiology, Amiloride/pharmacology, Animals, Body Fluids/*metabolism, Capillary Permeability, Dose-Response Relationship, Drug, Endothelium, Epithelial Cells/metabolism, Epithelial Sodium Channels, Epithelium/metabolism, Folkesson Hans G, Inhibitory Concentration 50, Li Tianbo, Lung/enzymology/*metabolism, Male, Messenger/antagonists & inhibitors/metabolism, Permeability, Plasmids/administration & dosage/pharmacology, Rats, RNA, Small Interfering/genetics/pharmacology, Sodium Channels/drug effects/genetics/metabolism/*physiology, Sprague-Dawley, Terbutaline/pharmacology, Tissue Distribution, Vascular/metabolism
Myocardial work load is a major determinant of norepinephrine-induced left ventricular dysfunction.
Tags: 1994, Allman F D, Anesthesia, Animals, Blood Pressure/*drug effects, Bosso F J, Cardiovascular, Consciousness, Diastole/drug effects, Dose-Response Relationship, Drug, General, Heart Rate/*drug effects, Heart/drug effects/*physiology, Left/drug effects/*physiology, Models, Norepinephrine/*pharmacology, Pentobarbital, Pilati C F, Rabbits, Systole/drug effects, The American journal of physiology, Time Factors, Ventricular Function
Acute exercise enhances nitric oxide modulation of vascular response to phenylephrine.
Tags: *Physical Exertion, 1993, Animals, Arginine/analogs & derivatives/pharmacology, Blood Flow Velocity, Blood Pressure/drug effects, Blood Vessels/*drug effects, Collins H L, DiCarlo S E, Dose-Response Relationship, Drug, Female, Heart Rate/drug effects, Iliac Artery/drug effects/physiology, Male, NG-Nitroarginine Methyl Ester, Nitric Oxide/antagonists & inhibitors/*physiology, Patil R D, Phenylephrine/*pharmacology, Rats, Sprague-Dawley, The American journal of physiology, Time Factors, Vasoconstriction/drug effects/physiology
Sexual dimorphism in vasopressin-induced contraction of rat aorta.
Endothelin-mediated in vivo pressor responses following TRPV1 activation.
Tags: *Blood Pressure/drug effects, *Vasoconstriction/drug effects, 2011, Adrenergic alpha-Agonists/administration & dosage, American journal of physiology. Heart and circulatory physiology, Analysis of Variance, Animal, Animals, Azepines/administration & dosage, Biphenyl Compounds/administration & dosage, Bratz Ian N, Capsaicin/administration & dosage, Cells, Cultured, Damron Derek S, Department of Integrative Medical Sciences, Diabetes Mellitus, Diabetic Angiopathies/genetics/*metabolism/physiopathology, Dipeptides/administration & dosage, Disease Models, Dose-Response Relationship, Drug, Endothelial Cells/metabolism, Endothelin A Receptor Antagonists, Endothelin A/metabolism, Endothelin B Receptor Antagonists, Endothelin B/metabolism, Endothelin-1/*metabolism, Enzyme-Linked Immunosorbent Assay, Femoral Artery/drug effects/*metabolism/physiopathology, Guarini Giacinta, Haney Rebecca M, Inbred C57BL, Indoles/administration & dosage, Infusions, Intravenous, Knockout, Male, Meszaros J Gary, Mice, NEOMED College of Medicine, Ohanyan Vahagn A, Phenylephrine/administration & dosage, Raman Priya, Receptor, Talasila Phani K, Thodeti Charles K, TRPV Cation Channels/agonists/deficiency/genetics/*metabolism, Type 2/genetics/*metabolism/physiopathology, Vasoconstrictor Agents/administration & dosage
Functional selectivity of NK1 receptor signaling: peptide agonists can preferentially produce receptor activation or desensitization.
Tags: 2006, Animals, CHO Cells, Cricetinae, Dose-Response Relationship, Drug, Humans, Neurokinin-1/agonists/drug effects/*physiology, Rana catesbeiana, Rats, Receptors, Signal Transduction/*physiology, Simmons Mark A, Substance P/metabolism/pharmacology, Tachykinins/metabolism/pharmacology, The Journal of pharmacology and experimental therapeutics
Activation of metabotropic glutamate receptor 1 dimers requires glutamate binding in both subunits.
Tags: 2005, Blotting, Calcium Channels/drug effects/metabolism, Department of Integrative Medical Sciences, DNA/biosynthesis/genetics, Dose-Response Relationship, Drug, Fluorescent Antibody Technique, Genes, Glutamic Acid/*metabolism, Humans, Kammermeier Paul J, Membrane Potentials/drug effects, Metabotropic Glutamate/genetics/*metabolism, myc/genetics, NEOMED College of Medicine, Patch-Clamp Techniques, Plasmids/genetics, Receptors, Signal Transduction/drug effects, Superior Cervical Ganglion/cytology/drug effects/metabolism, Sympathetic Nervous System/cytology/drug effects/metabolism, The Journal of pharmacology and experimental therapeutics, Western, Yun June
Evaluation of factors associated with achieving glycemic control in a pharmacist-managed diabetes clinic.
Tags: 2014, Ambulatory Care, Ambulatory Care/organization & administration, American journal of therapeutics, Blood Glucose – Drug Effects, Blood Glucose/drug effects, Boros Melanie L, Department of Internal Medicine, Department of Pharmaceutical Sciences, Department of Pharmacy Practice, Diabetes Mellitus, Dose-Response Relationship, Drug, Female, Follow-Up Studies, Frazee Lawrence A, Glycated Hemoglobin A/metabolism, Glycosylated – Metabolism, Hemoglobin A, Human, Humans, Hypoglycemic Agents – Administration and Dosage, Hypoglycemic Agents – Therapeutic Use, Hypoglycemic Agents/administration & dosage/*therapeutic use, Insulin – Administration and Dosage, Insulin – Therapeutic Use, Insulin/administration & dosage/therapeutic use, Kostoff Matthew D, Male, Middle Age, Middle Aged, Moorman John M, NEOMED College of Medicine, NEOMED College of Pharmacy, Pharmaceutical Services/*organization & administration, Pharmacists – Administration, Pharmacists/*organization & administration, Pharmacy Service – Administration, Prospective Studies, Retrospective Design, Retrospective Studies, Social Work – Statistics and Numerical Data, Social Work/statistics & numerical data, Treatment Outcome, Treatment Outcomes, Type 2 – Drug Therapy, Type 2/*drug therapy
Pyrethroid Insecticides Directly Activate Microglia Through Interaction With Voltage-Gated Sodium Channels.
Tags: *deltamethrin, *intracellular sodium., *Microglia, *neurodegeneration, *Neuroinflammation, *permethrin, *pyrethroids, *tetrodotoxin, *tumor necrosis factor, *Voltage-gated sodium channels, 2017, Animals, Cell Line, Department of Pharmaceutical Sciences, Dose-Response Relationship, Drug, Hossain Muhammad M, Inbred C57BL, Insecticides/*toxicity, Ion Channel Gating/*drug effects, Liu Jason, Mice, Microglia/*drug effects/metabolism, NEOMED College of Pharmacy, Pyrethrins/*toxicity, Richardson Jason R, Sodium Channels/*drug effects, Toxicological sciences : an official journal of the Society of Toxicology, Transformed, Tumor Necrosis Factor-alpha/metabolism
Selective Targeting of Heme Protein in Cytochrome P450 and Nitric Oxide Synthase by Diphenyleneiodonium.
Tags: *cytochrome P450, *flavoenzymes, *heme, *nitric oxide synthase, *Reactive oxygen species, 2016, Aleksunes Lauren M, Animals, Cytochrome P-450 Enzyme Inhibitors/*pharmacology, Cytochrome P-450 Enzyme System/*metabolism, Department of Pharmaceutical Sciences, Dose-Response Relationship, Drug, Heck Diane E, Heindel Ned D, Heme/*antagonists & inhibitors/metabolism, Humans, Jan Yi-Hua, Laskin Debra L, Laskin Jeffrey D, Liver/drug effects/enzymology, Mice, Microsomes, Mishin Vladimir, NEOMED College of Pharmacy, Nitric Oxide Synthase Type II/*antagonists & inhibitors/metabolism, Nitric Oxide/metabolism, Onium Compounds/*pharmacology, Rats, Recombinant Proteins/metabolism, Richardson Jason R, Sprague-Dawley, Szilagyi John T, Time Factors, Toxicological sciences : an official journal of the Society of Toxicology
Resveratrol inhibition of Propionibacterium acnes.
Tags: *Anti-Bacterial Agents, 2007, Anti-Inflammatory Agents, Bailey Erin, Benzoyl Peroxide/pharmacology, Booth Tristan D, Department of Family & Community Medicine, Docherty John J, Dose-Response Relationship, Drug, Erythromycin/pharmacology, Keratolytic Agents/pharmacology, McEwen Heather A, Microbial Sensitivity Tests, NEOMED College of Medicine, Non-Steroidal/*pharmacology, Propionibacterium acnes/*drug effects/growth & development, Resveratrol, Stilbenes/*pharmacology, Sweet Thomas J, The Journal of antimicrobial chemotherapy
Associations between Difficulty Paying Medical Bills and Forgone Medical and Prescription Drug Care.
Tags: *Fees, *Health Expenditures, *Health Services Accessibility, *Patient Compliance, *Prescription Fees, 2015, Adult, Aged, Baughman Kristin R, Bisexuals, Burke Ryan C, Cross-Sectional Studies, debt, Department of Family & Community Medicine, Drug, Family Health, Female, Financial, Health Status, Health Surveys, Hewit Michael S, Homeless Persons, Hull Sharon K, Humans, Male, Medical, Meeker James, Middle Aged, NEOMED College of Medicine, Ohio, Population Characteristics, Population health management, Prescriptions, Socioeconomic Factors, Special Populations, Sudano Joseph J, Young Adult
Secure cranial-mount intrathecal cannulation - a spinal administration technique in the rat.
Tags: 2000, Analgesics, Anesthesia, Animals, Crisp T, Dose-Response Relationship, Drug, Injections, Journal of neuroscience methods, Microinjections, Morphine/administration & dosage/pharmacology, Opioid/administration & dosage/pharmacology, Rats, Schechter J B, Spinal Cord/*physiology, Spinal/*instrumentation, Sprague-Dawley, Stereotaxic Techniques/*instrumentation
MDMA-like stimulus effects of hallucinogens in male Fawn-Hooded rats.
Tags: 1998, 4-methylenedioxyamphetamine/*pharmacology, Animals, Central Nervous System Stimulants/*pharmacology, Conditioning, Cues, Discrimination (Psychology)/drug effects, Dopamine Agents/pharmacology, Dose-Response Relationship, Drug, Generalization, Hallucinogens/*pharmacology, Inbred Strains, Male, N-Methyl-3, Operant/drug effects, Pharmacology, biochemistry, and behavior, Rats, Schechter M D, Serotonin Agents/pharmacology, Serotonin/genetics/physiology, Sprague-Dawley, Stimulus/drug effects
Rohypnol ("roofies") control of drug discrimination: effect of coadministered ethanol or flumenazil.
Tags: 1998, Animals, Anti-Anxiety Agents/*pharmacology, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Drug Administration Schedule, Ethanol/*pharmacology, Flumazenil/*pharmacology, Flunitrazepam/*pharmacology, GABA Antagonists/*pharmacology, Male, Pharmacology, biochemistry, and behavior, Rats, Schechter M D, Sprague-Dawley
Discriminative characteristics of high and low cocaine administration: effect of other psychostimulants.
Tags: 1997, Amphetamine/pharmacology, Animals, Central Nervous System Stimulants/pharmacology, Cocaine/*pharmacology, Conditioning, Discrimination Learning/*drug effects, Dopamine Agents/*pharmacology, Dose-Response Relationship, Drug, Drug Evaluation, Generalization, Male, Methamphetamine/pharmacology, Operant/*drug effects, Pharmacology, biochemistry, and behavior, Preclinical, Propiophenones/pharmacology, Psychotropic Drugs/*pharmacology, Rats, Response/*drug effects, Schechter M D
Drug-drug discrimination: stimulus properties of drugs of abuse upon a serotonergic-dopaminergic continuum.
Tags: 1997, 4-methylenedioxyamphetamine/pharmacology, Amphetamine/pharmacology, Animals, Discrimination (Psychology)/*drug effects, Dopamine Agonists/pharmacology, Dopamine Uptake Inhibitors/pharmacology, Dopamine/*physiology, Dose-Response Relationship, Drug, Generalization, Lysergic Acid Diethylamide/pharmacology, Male, N-Methyl-3, Norfenfluramine/pharmacology, Pharmacology, biochemistry, and behavior, Propiophenones/pharmacology, Rats, Schechter M D, Serotonin Agents/pharmacology, Serotonin Receptor Agonists/pharmacology, Serotonin Uptake Inhibitors/pharmacology, Serotonin/*physiology, Stimulus, Substance-Related Disorders/*psychology, Tetrahydronaphthalenes/pharmacology, Time Factors
Serotonergic mediation of fenfluramine discriminative stimuli in fawn-hooded rats.
Tags: *Discrimination Learning, 1997, 4-methylenedioxyamphetamine/pharmacology, Animals, Dose-Response Relationship, Drug, Fenfluramine/administration & dosage/*pharmacology, Fluoxetine/pharmacology, Ibogaine/pharmacology, Life sciences, Male, Methoxydimethyltryptamines/pharmacology, N-Methyl-3, Piperazines/pharmacology, Quipazine/pharmacology, Rats, Schechter M D, Serotonin Agents/administration & dosage/*pharmacology, Serotonin Receptor Agonists/pharmacology, Serotonin/*metabolism, Sprague-Dawley
Phentermine+fenfluramine produce cocaine-like discriminative cues.
Tags: *Discrimination (Psychology), 1996, Animals, Cocaine/*pharmacology, Department of Anatomy & Neurobiology, Dose-Response Relationship, Drug, Fenfluramine/administration & dosage/*pharmacology, Life sciences, Male, McBurney D, NEOMED College of Medicine, Phentermine/administration & dosage/*pharmacology, Rats, Schechter M D, Sprague-Dawley
Sex differences in extracellular and intracellular calcium-mediated vascular reactivity to vasopressin in rat aorta.
Tags: *Sex Characteristics, 1, 1998, 3-Pyridinecarboxylic acid, 4-dihydro-2, 6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Animals, Aorta/drug effects/*metabolism, Calcium Channel Agonists/*pharmacology, Calcium Channel Blockers/*pharmacology, Calcium/*metabolism, Department of Internal Medicine, Diltiazem/pharmacology, Dose-Response Relationship, Drug, Eatman D, European journal of pharmacology, Female, In Vitro Techniques, Male, Methyl ester/pharmacology, NEOMED College of Medicine, Potassium Chloride/pharmacology, Rats, Rutecki G W, Simvastatin/pharmacology, Sprague-Dawley, Stallone J N, Vasoconstriction/*drug effects, Vasopressins/*metabolism, Whittier F C
Discrete versus cumulative dosing in dose-response discrimination studies.
Tags: 1997, 4-methylenedioxyamphetamine/*pharmacology, Animals, Chemical, Cocaine/*pharmacology, Discrimination Learning/*drug effects, Dose-Response Relationship, Drug, Drug Administration Schedule, Drug Evaluation, European journal of pharmacology, Male, N-Methyl-3, Preclinical, Rats, Schechter M D, Sprague-Dawley, Stimulation
The effects of nicotine on dopamine and DOPAC output from rat striatal tissue.
Tags: 1998, 3, 4-Dihydroxyphenylacetic Acid/*metabolism, Amphetamine/pharmacology, Anderson L I, Animals, Central Nervous System Stimulants/pharmacology, Corpus Striatum/*drug effects/*metabolism, Dluzen D E, Dopamine/*metabolism, Dose-Response Relationship, Drug, European journal of pharmacology, Ganglionic Stimulants/administration & dosage/*pharmacology, Male, Nicotine/administration & dosage/*pharmacology, Potassium Chloride/pharmacology, Rats, Sprague-Dawley
Olanzapine attenuates the reinforcing effects of cocaine.
Tags: 1997, Animal/*drug effects, Animals, Antipsychotic Agents/administration & dosage/*pharmacology, Behavior, Benzodiazepines, Cocaine/administration & dosage/antagonists & inhibitors/*pharmacology, Conditioning, Dopamine Uptake Inhibitors/administration & dosage/*pharmacology, Dose-Response Relationship, Drug, European journal of pharmacology, Food Preferences/drug effects, Male, Meil W M, Olanzapine, Operant/*drug effects, Pirenzepine/administration & dosage/*analogs & derivatives/pharmacology, Rats, Schechter M D, Self Administration, Sprague-Dawley
Discrimination of cocaethylene in rats trained to discriminate between its components.
A subtherapeutic international normalized ratio despite increasing doses of warfarin: could this be malabsorption?
Tags: *Drug Resistance, 2000, Administration, Adult, Anticoagulants/administration & dosage/metabolism/pharmacokinetics/therapeutic use, Area Under Curve, Biological Availability, Delgado L L, Department of Family & Community Medicine, Department of Internal Medicine, Dose-Response Relationship, Drug, Female, Frazee L A, Haupt K M, Humans, Injections, Intestinal Absorption/*physiology, Intravenous, Kidney Transplantation, Lara L F, NEOMED College of Medicine, Oral, Rutecki G W, The American journal of the medical sciences, Warfarin/*administration & dosage/*metabolism/pharmacokinetics/therapeutic use
Localization and function of NK(3) subtype tachykinin receptors of layer V pyramidal neurons of the guinea-pig medial prefrontal cortex.
Tags: 2008, Animals, Autoradiography/methods, Dose-Response Relationship, Drug, Drug Interactions, Excitatory Amino Acid Antagonists/pharmacology, Excitatory Postsynaptic Potentials/drug effects/radiation effects, Guinea Pigs, In Vitro Techniques, Iodine Isotopes/pharmacokinetics, Male, Medd A M, Membrane Potentials/drug effects/physiology/radiation effects, Neurokinin B/analogs & derivatives/pharmacokinetics, Neurokinin-3/agonists/antagonists & inhibitors/*metabolism, Neuroscience, Patch-Clamp Techniques, Peptide Fragments/pharmacology, Prefrontal Cortex/*cytology, Protein Binding/drug effects, Pyramidal Cells/drug effects/*metabolism, Quinolines/pharmacology, Quinoxalines/pharmacology, Receptors, Simmons M A, Sobotka-Briner C D, Substance P/analogs & derivatives/pharmacology, Valine/analogs & derivatives/pharmacology
Valproate increases dopamine transporter expression through histone acetylation and enhanced promoter binding of Nurr1.
Tags: 2017, Acetylation/drug effects, Animals, Butyrates/pharmacology, Cell Line, Cell Survival/drug effects, Department of Pharmaceutical Sciences, Dopamine Plasma Membrane Transport Proteins/*metabolism, Dopamine transporter, Dopaminergic Neurons/cytology/drug effects/metabolism, Dose-Response Relationship, Drug, Eid Aseel, Epigenesis, Epigenetics, Genetic, Genetic/drug effects, Green Ashley L, Group A, Guo Grace L, HDAC, Histone deacetylase, Histone Deacetylase Inhibitors/*pharmacology, Histone Deacetylases/metabolism, Histones/*drug effects/metabolism, Homeodomain Proteins/metabolism, Hydroxamic Acids/pharmacology, Member 2/*metabolism, Messenger/metabolism, NEOMED College of Pharmacy, Neuropharmacology, Nuclear Receptor Subfamily 4, Nurr1, Pitx3, Promoter Regions, Rats, Richardson Jason R, RNA, Transcription Factors/metabolism, Valproate, Valproic Acid/*pharmacology, Zarbl Helmut, Zhan Le
Testosterone enhances dopamine depletion by methamphetamine in male, but not female, mice.
Tags: *Sex Characteristics, 2008, Animals, Castration/methods, Corpus Striatum/drug effects/metabolism, Dluzen Dean E, Dopamine Uptake Inhibitors/*pharmacology, Dopamine/*metabolism, Dose-Response Relationship, Drug, Female, Lewis Chandani, Male, Methamphetamine/*pharmacology, Mice, Neuroscience letters, Testosterone Propionate/*pharmacology
The effect of gender and the neurotrophin, BDNF, upon methamphetamine-induced neurotoxicity of the nigrostriatal dopaminergic system in mice.
Tags: 2004, Animals, Brain-Derived Neurotrophic Factor/deficiency/genetics/*metabolism, Central Nervous System Stimulants/poisoning, Corpus Striatum/*drug effects/*metabolism, Dluzen Dean E, Dopamine/*metabolism, Dose-Response Relationship, Drug, Female, Humans, Male, Methamphetamine/*poisoning, Mice, Mutation, Neuroscience letters, Neurotoxicity Syndromes/*etiology/*metabolism, Sex Factors, Structure-Activity Relationship, Substantia Nigra/drug effects/metabolism, Transgenic
The role of the N-terminal and mid-region residues of substance P in regulating functional selectivity at the tachykinin NK1 receptor.
Tags: 2008, Amino Acid Sequence, Animals, Beard Debbie J, Binding, Calcium Signaling/physiology, CHO Cells, Competitive/drug effects, Cricetinae, Cricetulus, Dose-Response Relationship, Drug, European journal of pharmacology, Iodine Radioisotopes, Ligands, Models, Molecular, Molecular Sequence Data, Neurokinin-1/chemistry/drug effects/*metabolism, Perrine Shane A, Rats, Receptors, Simmons Mark A, Substance P/chemistry/drug effects/*physiology, Young John K