Browse Items (215 total)
- Tags: Receptors
Orphan nuclear receptor oestrogen-related receptor gamma (ERRgamma) plays a key role in hepatic cannabinoid receptor type 1-mediated induction of CYP7A1 gene expression.
Tags: 2015, Animals, bile acid, Bile Acids and Salts/metabolism, Cannabinoid, cannabinoid receptors, CB1/agonists/genetics/*metabolism, Cells, Chiang John Y L, Choi Hueng-Sik, Cholesterol 7-alpha-Hydroxylase/*biosynthesis/genetics, cholesterol 7alpha-hydroxylase (CYP7A1), Cultured, Cytoplasmic and Nuclear/metabolism, Department of Integrative Medical Sciences, Drug Inverse Agonism, Estrogen/genetics/*metabolism, Ethanol/pharmacology, Gene Expression, Genetic, Glycerides/pharmacology, GSK5182, HEK293 Cells, Hepatocytes/metabolism, Humans, Inbred C57BL, Jeong Won-Il, Kim Don-Kyu, Kim Seong Heon, Knockout, Lee Chul-Ho, Lee In-Kyu, Lee Ji-Min, Liver/*metabolism, Mice, NEOMED College of Medicine, oestrogen-related receptor gamma (ERRgamma), orphan nuclear receptor, Park Seung Bum, Promoter Regions, Rats, Receptor, Receptors, small heterodimer partner (SHP), Sprague-Dawley, The Biochemical journal, Transcription, Zhang Yaochen
Identification of novel pathways that control farnesoid X receptor-mediated hypocholesterolemia.
Tags: 2010, Absorption, Anderson Jody, Animals, Biological, Cell Line, Cholesterol/*metabolism, Class B/*genetics/metabolism, Coronary Disease/metabolism, Cytoplasmic and Nuclear/*metabolism, Department of Integrative Medical Sciences, Edwards Peter A, Glucose/metabolism, Gonzalez Frank J, Hepatocyte Nuclear Factor 4/metabolism, Homeostasis, Humans, Lipoproteins/metabolism, Liver/metabolism, Ma Huiyan, Mice, Models, NEOMED College of Medicine, Receptors, Scavenger Receptors, The Journal of biological chemistry, Willson Timothy M, Yin Liya, Zhang Yanqiao
Loss of FXR protects against diet-induced obesity and accelerates liver carcinogenesis in ob/ob mice.
Tags: 2012, Adipose Tissue, Adiposity/genetics, Animals, Brown/pathology, Carcinoma/etiology/*genetics, Cell Transformation, Chen Wei-Dong, Cytoplasmic and Nuclear/*deficiency/genetics, Diet, Dietary Fats/metabolism, Edwards Peter A, Energy Metabolism/genetics, Female, Ge Xuemei, Gene Knockout Techniques, Glucose Intolerance/complications/genetics, Heemstra Lydia A, High-Fat/*adverse effects, Intestinal Absorption, Kasim Neda, Knockout, Leptin/deficiency/genetics, Liver Neoplasms/etiology/*genetics, Liver/pathology, Ma Huiyan, Male, Mice, Molecular endocrinology (Baltimore, Md.), Muscle, Neoplastic/genetics, Novak Colleen M, Obese, Obesity/*etiology/genetics, Receptors, Sex Factors, Skeletal/metabolism, Smith Joseph L, Weight Gain/genetics, Xu Jiesi, Zhang Yanqiao
Promoter activity and regulation of the CYP4F2 leukotriene B(4) omega-hydroxylase gene by peroxisomal proliferators and retinoic acid in HepG2 cells.
Tags: *Gene Expression Regulation, *Promoter Regions, 2000, Amino Acid Sequence, Archives of biochemistry and biophysics, Base Sequence, Cell Line, Chen L, Cloning, Cytochrome P-450 CYP4A, Cytochrome P-450 Enzyme System/*genetics/metabolism, Cytochrome P450 Family 4, Cytoplasmic and Nuclear/metabolism, Department of Integrative Medical Sciences, DNA, DNA Footprinting, Enzymologic, Exons, Genes, Genetic, Genetic/drug effects, Hardwick J P, Humans, Introns, Leukotriene B4/metabolism, Mixed Function Oxygenases/metabolism, Models, Molecular, Molecular Sequence Data, NEOMED College of Medicine, Peroxisome Proliferators/*metabolism, Receptors, Reporter, Retinoic Acid Receptor alpha, Retinoic Acid/metabolism, Sequence Analysis, Transcription, Transcription Factors/metabolism, Transfection, Tretinoin/*metabolism, Zhang X
Transcriptional regulation of the human sterol 12alpha-hydroxylase gene (CYP8B1): roles of heaptocyte nuclear factor 4alpha in mediating bile acid repression.
Tags: *DNA-Binding Proteins, *Transcription, 2001, Base Sequence, Basic Helix-Loop-Helix Leucine Zipper Transcription Factors, Bile Acids and Salts/*pharmacology, Binding Sites, Chiang J Y, Cholesterol 7-alpha-Hydroxylase/genetics, Cultured, Cytochrome P-450 Enzyme System/*genetics, Cytoplasmic and Nuclear/physiology, Department of Integrative Medical Sciences, Genetic, Genetic/physiology, Hepatocyte Nuclear Factor 4, Humans, Molecular Sequence Data, NEOMED College of Medicine, Phosphoproteins/*physiology, Promoter Regions, Receptors, Repressor Proteins/*pharmacology, Steroid 12-alpha-Hydroxylase, Steroid Hydroxylases/*genetics, The Journal of biological chemistry, Transcription Factors/*physiology, Tumor Cells, Zhang M
Synthesis and biological evaluations of chalcones, flavones and chromenes as farnesoid x receptor (FXR) antagonists.
Tags: 2017, Animals, Antagonist, Benzopyrans/chemical synthesis/*pharmacology, Chalcones, Chalcones/chemical synthesis/*pharmacology, Chen Yuan, Chromenes, Cytoplasmic and Nuclear/*antagonists & inhibitors, Deng Ruitang, European journal of medicinal chemistry, Fang Weishuo, Farnesoid X receptor, Flavones/chemical synthesis/*pharmacology, Huan Yi, Jiang Qian, Liu Jinsong, Liu Shuainan, Liver Diseases/drug therapy, Liver/chemistry/*drug effects/metabolism, Mice, Receptors, Shen Zhufang, Sun Deyang, Tan Wenjuan, Triglycerides/analysis, Verma Ruchi, Wang Na, Wang Xing, Wong Chiwai, Xu Yang, Zhang Guoning, Zhang Yanqiao
Stimulation of distal airspace fluid clearance in guinea pigs involves bumetanide-sensitive ion transport.
Tags: *Ion Transport, 2004, Absorption, Adrenergic, Adrenergic beta-Antagonists/pharmacology, American journal of obstetrics and gynecology, Animals, beta/physiology, Body Fluids/*metabolism, Bumetanide/*pharmacology, Diuretics/*pharmacology, Epinephrine/blood, Epithelium, Fetus/metabolism, Folkesson Hans G, Gestational Age, Guinea Pigs, Lung/*embryology/metabolism, Newborn, Norlin Andreas, Propranolol/pharmacology, Receptors, Ye Xin
A neurochemical heterogeneity of the rat striatum as measured by in vivo electrochemistry and microdialysis.
Tags: 1990, 3, 4-Dihydroxyphenylacetic Acid/metabolism, Amphetamines/*pharmacology, Animals, Brain research, Corpus Striatum/*metabolism, Dopamine D2, Dopamine/*metabolism, Dopamine/drug effects, Electrochemistry, Inbred Strains, Male, Pehek E A, Rats, Receptors, Sulpiride/*pharmacology, Yamamoto B K
A metabolic stress-inducible miR-34a-HNF4alpha pathway regulates lipid and lipoprotein metabolism.
Tags: 2015, Animals, Apolipoproteins E/genetics, Atherosclerosis/genetics/metabolism, Department of Integrative Medical Sciences, Diabetes Mellitus, Experimental/genetics/metabolism, Hep G2 Cells, Hepatocyte Nuclear Factor 4/*genetics/metabolism, Humans, Knockout, LDL/genetics, Li Yuanyuan, Lipid Metabolism/*genetics, Lipoproteins/metabolism, Liver/metabolism, Mice, MicroRNAs/*genetics/metabolism, Middle Aged, Nature communications, NEOMED College of Medicine, Non-alcoholic Fatty Liver Disease/*genetics/metabolism, Physiological/*genetics, Receptors, Stress, Triglycerides/*metabolism, Xu Jiesi, Xu Yang, Yin Liya, Zalzala Munaf, Zhang Yanqiao
Farnesoid X receptor activation increases reverse cholesterol transport by modulating bile acid composition and cholesterol absorption in mice.
Tags: *Intestinal Absorption, 2016, Adorini Luciano, Animals, Bile Acids and Salts/*chemistry, Biological Transport, Cholesterol/*metabolism, Cytoplasmic and Nuclear/*physiology, Department of Integrative Medical Sciences, Gonzalez Frank J, Hepatology (Baltimore, Md.), Inbred C57BL, Lee Yoon-Kwang, Li Fei, Mice, NEOMED College of Medicine, Receptors, Xu Jiesi, Xu Yang, Yin Liya, Zalzala Munaf, Zhang Yanqiao
Hepatic carboxylesterase 1 is essential for both normal and farnesoid X receptor-controlled lipid homeostasis.
Tags: *Homeostasis, *Lipid Metabolism, 2014, Adorini Luciano, Animals, Carboxylic Ester Hydrolases/*physiology, Chen Wei-Dong, Cholesterol/blood, Cytoplasmic and Nuclear/*physiology, Department of Integrative Medical Sciences, Fatty Acids/metabolism, Ge Xuemei, Hepatology (Baltimore, Md.), Inbred C57BL, Jadhav Kavita, Li Yuanyuan, Lipogenesis, Liver/*enzymology, Mice, NEOMED College of Medicine, Receptors, Sterol Regulatory Element Binding Protein 1/physiology, Triglycerides/metabolism, Xu Jiesi, Xu Yang, Yin Liya, Zhang Yanqiao
Synaptic activity-induced Ca(2+) signaling in avian cochlear nucleus magnocellularis neurons.
Tags: 2012, Animals, Calcium Signaling/*physiology, Chick Embryo, Chickens, Cochlear Nucleus/*metabolism, Department of Anatomy & Neurobiology, GABA-A/metabolism, Inhibitory Postsynaptic Potentials/physiology, Lu Yong, NEOMED College of Medicine, Neurons/*metabolism, Neuroscience research, Organ Culture Techniques, Patch-Clamp Techniques, Receptors, Synapses/*metabolism, Synaptic Transmission/*physiology, Tang Zheng-Quan, Wang Lie-Cheng
Transcriptional regulation of the human cholesterol 7 alpha-hydroxylase gene (CYP7A) in HepG2 cells.
Tags: *Promoter Regions, *Transcription, *Transcription Factors, 1996, Base Sequence, Binding Sites, Cell Line, Chiang J Y, Cholesterol 7-alpha-Hydroxylase/biosynthesis/*genetics, Consensus Sequence, Crestani M, Department of Integrative Medical Sciences, DNA-Binding Proteins/genetics/metabolism, Enzyme Repression, Enzymologic/*drug effects, Galli G, Gene Expression Regulation, Genes, Genetic, Glucocorticoid/genetics/metabolism, Glucocorticoids/pharmacology, Hepatocyte Nuclear Factor 3-alpha, Humans, Insulin/pharmacology, Journal of lipid research, Marrapodi M, Molecular Sequence Data, NEOMED College of Medicine, Nuclear Proteins/genetics/metabolism, Phorbol Esters/pharmacology, Receptors, Recombinant Fusion Proteins/biosynthesis, Reporter, Stroup D, Thyroid Hormones/pharmacology, Transfection, Wang D P
Comparison of inotropic and chronotropic effects of vasoactive intestinal peptide in isolated dog atria
Tags: 1996, adenylate-cyclase, anesthetized dogs, atrium, autonomic nervous system, Cardiac, conscious dogs, contractile force, Heart Rate, isoproterenol, Journal Article, Journal of the Autonomic Nervous System, neuropeptide, neuropeptides, Neurosciences & Neurology, parasympathetic, Performance, polypeptide, Receptor, Receptors, Stuesse S L, SUBSTANCE P, VIP, Wallick D W
mGluRs modulate neuronal firing in the auditory midbrain.
Tags: 2011, Acoustic Stimulation/methods, Action Potentials/drug effects/*physiology, Animals, Auditory Perception/drug effects/physiology, Department of Anatomy & Neurobiology, Excitatory Amino Acid Agonists/pharmacology, Excitatory Amino Acid Antagonists/pharmacology, Galazyuk A V, Glutamic Acid/physiology, Inbred CBA, Inferior Colliculi/drug effects/metabolism/*physiology, Metabotropic Glutamate/agonists/antagonists & inhibitors/*physiology, Mice, NEOMED College of Medicine, Neural Inhibition/drug effects/physiology, Neurons/drug effects/*physiology, Neuroscience letters, Perceptual Masking/physiology, Receptors, Synaptic Transmission/drug effects/physiology, Voytenko S V
Ontogenesis of the depressant activity of carbachol on synaptic activity in rat visual cortex.
Efficacy and safety of ustekinumab and etanercept for the treatment of psoriasis.
Tags: 2010, Anti-Inflammatory Agents/adverse effects/*therapeutic use, Antibodies, Etanercept, Evidence-Based Medicine, Expert opinion on biological therapy, Feldman Steven R, Humanized, Humans, Immunoglobulin G/adverse effects/*therapeutic use, Immunosuppressive Agents/adverse effects/*therapeutic use, Monoclonal, Monoclonal/adverse effects/*therapeutic use, Patient Selection, Psoriasis/*drug therapy/immunology, Receptors, Risk Assessment, Severity of Illness Index, Treatment Outcome, Tumor Necrosis Factor/*therapeutic use, Uhlenhake Elizabeth E, Ustekinumab
The orphan nuclear receptor small heterodimer partner is required for thiazolidinedione effects in leptin-deficient mice.
Tags: 2015, Animals, Bile Acids and Salts/metabolism, Cytoplasmic and Nuclear/biosynthesis/*genetics/metabolism, Department of Integrative Medical Sciences, Diabetes Mellitus/*drug therapy/genetics/metabolism, Gene Expression Regulation/drug effects, Glucose/metabolism, Hepatocytes/drug effects, Humans, Insulin Resistance/genetics, Insulin/*metabolism, Journal of biomedical science, Lee Yoon-Kwang, Leptin/deficiency/genetics, Lipid Metabolism/drug effects, Messenger/genetics, Mice, Moore David D, NEOMED College of Medicine, Obese, Park Young Joo, PPAR gamma/*biosynthesis/genetics, Receptors, RNA, Thiazolidinediones/*administration & dosage, Tseng Hsiu-Ting
G protein coupling profile of mGluR6 and expression of G alpha proteins in retinal ON bipolar cells.
Tags: 2006, Animals, Calcium/metabolism, Gene Expression/drug effects/*physiology, Glutamic Acid/pharmacology, GTP-Binding Protein alpha Subunits/*metabolism, Kammermeier Paul J, Membrane Potentials/drug effects/physiology/radiation effects, Metabotropic Glutamate/*metabolism, Microinjections/methods, Patch-Clamp Techniques/methods, Pertussis Toxin/pharmacology, Propionates/pharmacology, Rats, Receptors, Retina/*cytology, Retinal Bipolar Cells/drug effects/*metabolism/radiation effects, Reverse Transcriptase Polymerase Chain Reaction/methods, Tian Liantian, Visual neuroscience, Wistar
Synaptic plasticity in the hippocampal slice: functional consequences.
Comparative aspects of hippocampal and neocortical long-term potentiation.
Development of GPCR modulation of GABAergic transmission in chicken nucleus laminaris neurons.
Tags: *Synaptic Transmission, 2012, Animals, Brain/*cytology, Chickens/*metabolism, Department of Anatomy & Neurobiology, G-Protein-Coupled/*metabolism, GABA-A/metabolism, GABA-B/metabolism, gamma-Aminobutyric Acid/*metabolism, Lu Yong, Metabotropic Glutamate/metabolism, NEOMED College of Medicine, Neurons/*metabolism, Patch-Clamp Techniques, PloS one, Receptors, Synapses/metabolism, Tang Zheng-Quan
Two GABAA responses with distinct kinetics in a sound localization circuit.
Tags: *Sound, 2012, Animals, Chick Embryo, Chickens, Department of Anatomy & Neurobiology, Female, GABA-A/*physiology, gamma-Aminobutyric Acid/metabolism, Lu Yong, Male, NEOMED College of Medicine, Neurons/*metabolism, Pitch Discrimination, Receptors, Sound Localization/*physiology, Synapses/physiology, Tang Zheng-Quan, The Journal of physiology
Activation of synaptic group II metabotropic glutamate receptors induces long-term depression at GABAergic synapses in CNS neurons.
Tags: 2013, Amino Acids/pharmacology, Animals, Chick Embryo, Cochlear Nucleus/drug effects/metabolism, Curry Rebecca J, Cyclopropanes/pharmacology, Department of Anatomy & Neurobiology, Dinh Emilie Hoang, Excitatory Amino Acid Agonists/pharmacology, Excitatory Amino Acid Antagonists/pharmacology, Excitatory Postsynaptic Potentials/drug effects/physiology, GABAergic Neurons/drug effects/*metabolism, Glycine/analogs & derivatives/pharmacology, Hamlet William R, Inhibitory Postsynaptic Potentials/drug effects/physiology, Liu Yu-Wei, Long-Term Synaptic Depression/drug effects/*physiology, Lu Yong, Metabotropic Glutamate/agonists/antagonists & inhibitors/*metabolism, NEOMED College of Medicine, Neural Inhibition/drug effects/physiology, Receptors, Shi Wei, Synapses/drug effects/*metabolism, Synaptic Transmission/drug effects/*physiology, Tang Zheng-Quan, The Journal of neuroscience : the official journal of the Society for Neuroscience, Xanthenes/pharmacology
Ambient GABA-activated tonic inhibition sharpens auditory coincidence detection via a depolarizing shunting mechanism.
Tags: 2011, Animals, Auditory Pathways/*physiology, Blotting, Chick Embryo, Department of Anatomy & Neurobiology, Dinh Emilie Hoang, Electric Stimulation, GABA-A/*physiology, gamma-Aminobutyric Acid/*physiology, Inhibitory Postsynaptic Potentials, Lu Yong, Membrane Potentials/physiology, NEOMED College of Medicine, Neural Inhibition/*physiology, Neurons/*physiology, Patch-Clamp Techniques, Receptors, Shi Wei, Tang Zheng-Quan, The Journal of neuroscience : the official journal of the Society for Neuroscience, Western
Thermoreversible gel for delivery of activin receptor-like kinase 5 inhibitor
Tags: *Drug Delivery Systems, 2013, Animal, Animals, Benzodioxoles/*administration & dosage/pharmacokinetics/toxicity, Bhatia Deepak, Body Temperature, Delayed-Action Preparations, Disease Models, Drug Carriers/chemistry/toxicity, Fibroblasts/drug effects/metabolism, Filtering Surgery/*methods, Geldenhuys Werner, Gels, Glaucoma/*surgery, Imidazoles/*administration & dosage/pharmacokinetics/toxicity, Miladore Nicholas, Nakamura Hiroshi, Pharmaceutical development and technology, Poloxamer/chemistry/toxicity, Protein-Serine-Threonine Kinases/antagonists & inhibitors, Pyridines/*administration & dosage/pharmacokinetics/toxicity, Rabbits, Receptor, Receptors, Sutariya Vijaykumar, Temperature, Time Factors, Transforming Growth Factor beta/antagonists & inhibitors, Transforming Growth Factor-beta Type I, Viscosity, Wehrung Daniel
Orphan receptors chicken ovalbumin upstream promoter transcription factor II (COUP-TFII) and retinoid X receptor (RXR) activate and bind the rat cholesterol 7alpha-hydroxylase gene (CYP7A).
Tags: *Gene Expression Regulation, *Receptors, 1997, Animals, Chiang J Y, Chickens, Cholesterol 7-alpha-Hydroxylase/*genetics/metabolism, Circadian Rhythm, COUP Transcription Factor I, COUP Transcription Factor II, COUP Transcription Factors, Crestani M, Department of Integrative Medical Sciences, DNA-Binding Proteins/*metabolism, Electrophoresis, Enzymologic, Genetic, Glucocorticoid/*genetics, Models, Molecular, NEOMED College of Medicine, Nuclear Proteins/*metabolism, Polyacrylamide Gel, Promoter Regions, Rats, Receptors, Recombinant Proteins/genetics/metabolism, Retinoic Acid/*metabolism, Retinoid X Receptors, Steroid, Stroup D, The Journal of biological chemistry, Transcription Factors/*metabolism
HNF4 and COUP-TFII interact to modulate transcription of the cholesterol 7 alpha-hydroxylase gene (CYP7A1)
Tags: 2000, BILE acids, bile-acid synthesis, Biochemistry & Molecular Biology, Chiang J Y L, chicken ovalbumin, cholesterol metabolism, dna-binding, Hepatocyte Nuclear Factor 4, hormone-receptor superfamily, Journal Article, Journal of lipid research, messenger-rna, orphan receptors, promoter, Receptors, Response Elements, retinoic acid, Stroup D, thyroid-hormone, transcriptional regulation, upstream promoter transcription factor II
Acute and subchronic effects of methylenedioxymethamphetamine [(+/-)MDMA] on locomotion and serotonin syndrome behavior in the rat.
Tags: 1989, 3, 4-methylenedioxyamphetamine, 4-Methylenedioxyamphetamine/analogs & derivatives/*pharmacology, Amphetamines/*pharmacology, Animal/*drug effects, Animals, Behavior, Designer Drugs/*pharmacology, Dose-Response Relationship, Drug, Inbred Strains, Male, Motor Activity/*drug effects, N-Methyl-3, Pharmacology, biochemistry, and behavior, Rats, Receptors, Serotonin/*drug effects, Spanos L J, Time Factors, Yamamoto B K
A comparative analysis of monoaminergic involvement in the spinal antinociceptive action of DAMPGO and DPDPE.
Tags: 1989, 5)-, Ala(2)-MePhe(4)-Gly(5)-, Amines – Physiology, Anesthetics – Pharmacodynamics, Anesthetics/*pharmacology, Animals, Biogenic Monoamines/*physiology, Cell Surface – Drug Effects, Cell Surface – Physiology, Crisp T, D-Penicillamine (2, Dose-Response Relationship, Drug, Enkephalin, Enkephalins, Enkephalins – Pharmacodynamics, Enkephalins/*pharmacology, Inbred Strains, Injections, Intraspinal, Male, Naloxone – Pharmacodynamics, Naloxone/pharmacology, Opioid/drug effects/*physiology, Pain, Pain – Metabolism, Pain/*metabolism, Rats, Receptors, Spanos L J, Spinal, Spinal Cord – Drug Effects, Spinal Cord – Metabolism, Spinal Cord – Physiopathology, Spinal Cord/drug effects/metabolism/*physiopathology, Stafinsky J L
Bile acids activate fibroblast growth factor 19 signaling in human hepatocytes to inhibit cholesterol 7alpha-hydroxylase gene expression.
Tags: 2009, Butadienes/pharmacology, Carcinoma, Cell Line, Chenodeoxycholic Acid/*pharmacology, Chiang John Y L, Cholesterol 7-alpha-Hydroxylase/*biosynthesis, Cytoplasmic and Nuclear/metabolism/physiology, Department of Integrative Medical Sciences, DNA-Binding Proteins/metabolism, Fibroblast Growth Factor, Fibroblast Growth Factors/drug effects/*physiology, Gene Expression/drug effects, Hepatocellular/metabolism, Hepatocytes/metabolism, Hepatology (Baltimore, Md.), Humans, Isoxazoles/pharmacology, Li Tiangang, Mitogen-Activated Protein Kinase 1/metabolism, Mitogen-Activated Protein Kinase 3/metabolism, NEOMED College of Medicine, Nitriles/pharmacology, Owsley Erika, Receptor, Receptors, Signal Transduction/drug effects, Song Kwang-Hoon, Strom Stephen, Transcription Factors/metabolism, Tumor, Type 4/antagonists & inhibitors
Farnesoid X Receptor Activation by Obeticholic Acid Elevates Liver Low-Density Lipoprotein Receptor Expression by mRNA Stabilization and Reduces Plasma Low-Density Lipoprotein Cholesterol in Mice.
Functional selectivity, ligand-directed trafficking, conformation-specific agonism: what's in a name?
Functional selectivity of NK1 receptor signaling: peptide agonists can preferentially produce receptor activation or desensitization.
Tags: 2006, Animals, CHO Cells, Cricetinae, Dose-Response Relationship, Drug, Humans, Neurokinin-1/agonists/drug effects/*physiology, Rana catesbeiana, Rats, Receptors, Signal Transduction/*physiology, Simmons Mark A, Substance P/metabolism/pharmacology, Tachykinins/metabolism/pharmacology, The Journal of pharmacology and experimental therapeutics
Localization and function of NK(3) subtype tachykinin receptors of layer V pyramidal neurons of the guinea-pig medial prefrontal cortex.
Tags: 2008, Animals, Autoradiography/methods, Dose-Response Relationship, Drug, Drug Interactions, Excitatory Amino Acid Antagonists/pharmacology, Excitatory Postsynaptic Potentials/drug effects/radiation effects, Guinea Pigs, In Vitro Techniques, Iodine Isotopes/pharmacokinetics, Male, Medd A M, Membrane Potentials/drug effects/physiology/radiation effects, Neurokinin B/analogs & derivatives/pharmacokinetics, Neurokinin-3/agonists/antagonists & inhibitors/*metabolism, Neuroscience, Patch-Clamp Techniques, Peptide Fragments/pharmacology, Prefrontal Cortex/*cytology, Protein Binding/drug effects, Pyramidal Cells/drug effects/*metabolism, Quinolines/pharmacology, Quinoxalines/pharmacology, Receptors, Simmons M A, Sobotka-Briner C D, Substance P/analogs & derivatives/pharmacology, Valine/analogs & derivatives/pharmacology
The role of dopamine and serotonin receptors in the mediation of the ethanol interoceptive cue.
Tags: 1988, Animals, Conditioning, Cues, Discrimination (Psychology)/*physiology, Dopamine/drug effects/*physiology, Dose-Response Relationship, Drug, Ethanol/*pharmacology, Inbred Strains, Male, Operant/physiology, Pharmacology, biochemistry, and behavior, Rats, Receptors, Schechter M D, Serotonin/drug effects/*physiology, Signs S A
Metabotropic glutamate and GABA receptors modulate cellular excitability and glutamatergic transmission in chicken cochlear nucleus angularis neurons.
Tags: *Cellular excitability, *GABA(B)R, *mGluR, *Neuromodulation, *Nucleus angularis, *Synaptic Transmission, 2017, Action Potentials/drug effects, Animals, Chick Embryo, Cochlear Nucleus/cytology/*physiology, Department of Anatomy & Neurobiology, Excitatory Postsynaptic Potentials/drug effects, GABA-B Receptor Agonists/pharmacology, GABA-B/*physiology, Glutamic Acid/*physiology, Hearing research, Lu Yong, Metabotropic Glutamate/agonists/classification/*physiology, NEOMED College of Medicine, Neurons/drug effects/physiology, Patch-Clamp Techniques, Receptors, Shi Wei, Synaptic Transmission/drug effects
Nisoxetine infusion into the olfactory bulb enhances the capacity for male rats to identify conspecifics.
Tags: 2001, Adrenergic, Adrenergic alpha-Antagonists/pharmacology, alpha/drug effects/metabolism, Animal/*drug effects/physiology, Animal/drug effects/physiology, Animals, Behavior, Dluzen D E, Drug Interactions/physiology, Female, Fluoxetine/analogs & derivatives/*pharmacology, Hierarchy, Male, Neuroscience, Norepinephrine/*antagonists & inhibitors/metabolism, Olfactory Bulb/cytology/*drug effects/metabolism, Phentolamine/pharmacology, Presynaptic Terminals/drug effects/metabolism, Rats, Receptors, Recognition (Psychology)/*drug effects/physiology, Sexual Behavior, Shang Y, Smell/*drug effects/physiology, Social, Social Facilitation, Sprague-Dawley/anatomy & histology/*metabolism/psychology