Browse Items (215 total)
- Tags: Receptors
Effect of aging on the substance P receptor, NK-1, in the spinal cord of rats with peripheral nerve injury.
Tags: *Peripheral Nerve Injuries, 2001, Aging/*physiology, Animals, Computer-Assisted, Crisp T, Cruce W L, Hot Temperature, Image Processing, Immunohistochemistry, Inbred BN, Inbred F344, Lovell J A, Neurokinin-1/*metabolism, Rats, Receptors, Somatosensory & motor research, Spinal Cord/*metabolism, Stuesse S L, Thermosensing/physiology, Touch/physiology
Synaptic Inhibition in Avian Interaural Level Difference Sound Localizing Neurons.
Tags: *dorsal nucleus of the lateral lemniscus, *GABAA receptor, *interaural level difference, *reversal potential, *synaptic inhibition, 2016, Acoustic Stimulation/methods, Animals, Anions/metabolism, Avian Proteins/metabolism, Brain Stem/cytology/drug effects/*physiology, Chick Embryo, Chlorides/metabolism, Curry Rebecca J, Department of Anatomy & Neurobiology, Electric Stimulation, eNeuro, Female, GABA-A/metabolism, gamma-Aminobutyric Acid/metabolism, Glycine/metabolism, Intracellular Space/drug effects/metabolism, Lu Yong, Male, NEOMED College of Medicine, Neural Inhibition/drug effects/*physiology, Neurons/cytology/drug effects/*physiology, Patch-Clamp Techniques, Receptors, Sound Localization/drug effects/*physiology, Symporters/metabolism, Synaptic Transmission/drug effects/*physiology, Tissue Culture Techniques
Spermine depresses NMDA, K/AMPA and GABAA-mediated synaptic transmission in the rat hippocampal slice preparation.
Tags: 1994, AMPA/antagonists & inhibitors, Animals, Brain research, Calcium Channels/drug effects, DiScenna P G, Eterovic V A, Evoked Potentials/drug effects, Excitatory Amino Acid Antagonists/*pharmacology, Ferchmin P A, GABA-A Receptor Antagonists, Hippocampus/drug effects/*physiology, In Vitro Techniques, N-Methyl-D-Aspartate/antagonists & inhibitors, Rats, Receptors, Spermine/*pharmacology, Synapses/drug effects/*physiology, Synaptic Transmission/*drug effects, Teyler T J
The development of GABAB-mediated activity in the rat dentate gyrus.
Tags: 1994, Animals, Baclofen/analogs & derivatives/pharmacology, Brain research. Developmental brain research, DiScenna P G, Electric Stimulation, Evoked Potentials/drug effects, GABA-A Receptor Antagonists, GABA-A/drug effects/physiology, GABA-B Receptor Antagonists, GABA-B/*metabolism, Hippocampus/*growth & development/*metabolism, In Vitro Techniques, Nowicky A V, Organophosphorus Compounds/pharmacology, Rats, Receptors, Teyler T J
Oxytocin induces preservation of social recognition in male rats by activating alpha-adrenoceptors of the olfactory bulb.
Tags: *Social Behavior, 2000, Adrenergic, Adrenergic alpha-Agonists/pharmacology, Adrenergic alpha-Antagonists/pharmacology, Adrenergic beta-Agonists/pharmacology, Adrenergic beta-Antagonists/pharmacology, alpha/*drug effects/physiology, Animals, Clonidine/pharmacology, Dluzen D E, Ebner K, Engelmann M, Isoproterenol/pharmacology, Landgraf R, Male, Memory/*drug effects/physiology, Microdialysis, Muraoka S, Norepinephrine/pharmacology, Olfactory Bulb/*drug effects/physiology, Oxytocin/*pharmacology, Oxytocin/drug effects/*physiology, Phentolamine/pharmacology, Rats, Receptors, Social Dominance, The European journal of neuroscience, Timolol/pharmacology, Wistar
Unconventional effects of estrogen uncovered.
Tags: 2005, Animals, Corpus Striatum/*metabolism/physiology, Dluzen Dean E, Dopamine D2/metabolism, Dopamine/*metabolism, Estrogens/*physiology, GTP-Binding Proteins/metabolism, Humans, Receptors, Signal Transduction/physiology, Substantia Nigra/*metabolism/physiology, Trends in pharmacological sciences
Identification and functional characterization of two type VI collagen receptors, alpha 3 beta 1 integrin and NG2, during avian corneal stromal development.
Tags: 1998, Animals, Antigens/*metabolism, Birk D E, Cell Culture Techniques, Cell Movement/physiology, Cell Polarity/physiology, Cell Size/physiology, Chick Embryo, Collagen/*metabolism, Corneal Stroma/*embryology/*metabolism, Doane K J, Extracellular Matrix/metabolism, Fibroblasts/metabolism, Fluorescent Antibody Technique, Howell S J, Immunoblotting, Indirect, Integrin alpha3beta1, Integrins/*metabolism, Investigative ophthalmology & visual science, Laminin/*metabolism, Proteoglycans/*metabolism, Receptors
The contribution of interleukin-2 to effective wound healing.
Tags: *cutaneous diseases, *CYTOKINES, *immunotherapy, *Interleukin-2, *therapeutic targets, *Wound Healing, 2017, Animals, Cell Differentiation/physiology, Cell Proliferation/physiology, DelloStritto Daniel J, Diabetes Mellitus/metabolism/pathology, Doersch Karen M, Experimental biology and medicine (Maywood, N.J.), Humans, Interleukin-2/*metabolism, Interleukin-2/*metabolism/*therapeutic use, Lupus Erythematosus, Mice, Myocardial Infarction/metabolism/pathology, Newell-Rogers M Karen, Receptors, Sarcoidosis/metabolism/pathology, Signal Transduction/physiology, Skin/*injuries, Systemic/metabolism/pathology, T-Lymphocytes/cytology/immunology, Wound Healing/*physiology
G-protein-coupled bile acid receptor plays a key role in bile acid metabolism and fasting-induced hepatic steatosis in mice.
Tags: *Gene Expression Regulation, 2017, Analysis of Variance, Animal, Animals, Bile Acids and Salts/*metabolism, Boehme Shannon, Chiang John Y L, Department of Integrative Medical Sciences, Disease Models, Donepudi Ajay C, Energy Metabolism/physiology, Fasting, Fatty Liver/*metabolism/pathology, G-Protein-Coupled/*genetics, Hepatology (Baltimore, Md.), Homeostasis/genetics, Inbred C57BL, Li Feng, Lipid Metabolism/genetics, Male, Mice, NEOMED College of Medicine, Oxygen Consumption/physiology, Random Allocation, Receptors, RNA-Binding Proteins/*metabolism, Signal Transduction
Myocardial CXCR4 expression is required for mesenchymal stem cell mediated repair following acute myocardial infarction.
Tags: 2012, Agarwal U, Animal Studies, Apoptosis – Physiology, Cardiovascular System Physiology, Cell Movement – Physiology, Cell Physiology, Cell Surface, Cell Surface – Metabolism, Cells, Circulation, Coronary Circulation – Physiology, Cytokines – Metabolism, Department of Integrative Medical Sciences, Dong F, Finan A, Gene Expression – Physiology, Harvey J, Mice, myocardial infarction, Myocardial Infarction – Pathology, Myocardial Infarction – Therapy, Myocardium, NEOMED College of Medicine, Penn M S, Proteins, Receptors, Stem Cells – Metabolism, Stem Cells – Transplantation, Weber K
Myocardial CXCR4 expression is required for mesenchymal stem cell mediated repair following acute myocardial infarction.
Tags: 2012, Agarwal Udit, Animals, Apoptosis/physiology, Cardiac/cytology/physiology, Cell Movement/physiology, Chemokine CXCL12/*metabolism, Circulation, Coronary Circulation/physiology, CXCR4/*genetics/metabolism, Department of Integrative Medical Sciences, Dong Feng, Finan Amanda, Gene Expression/physiology, Green Fluorescent Proteins/genetics, Harvey James, Inbred C57BL, Knockout, Mesenchymal Stem Cell Transplantation/*methods, Mesenchymal Stem Cells/*metabolism, Mice, Myocardial Infarction/genetics/pathology/*therapy, Myocardium/cytology, Myocytes, NEOMED College of Medicine, Paracrine Communication/physiology, Penn Marc S, Receptors, Ventricular Remodeling/physiology, Weber Kristal
Cysteinyl leukotriene 2 receptor promotes endothelial permeability, tumor angiogenesis, and metastasis.
Tags: *angiogenesis, *cysteinyl leukotriene receptors, *endothelial cells, *metastasis, *tumor growth, 2019, Adapala Ravi K, Animals, Austen K Frank, Capillary Permeability/drug effects, Cyclohexanecarboxylic Acids/pharmacology, Department of Integrative Medical Sciences, Duah Ernest, Endothelial Cells/*drug effects, Experimental, Gene Knockout Techniques, Inbred C57BL, Kanaoka Yoshihide, Keshamouni Venkateshwar G, Kondeti Vinay, Leukotriene Antagonists/pharmacology, Leukotriene/drug effects/*metabolism, Lung Neoplasms/drug therapy, Male, Mice, NEOMED College of Medicine, Neoplasm Metastasis/drug therapy, Neoplasm Transplantation, Neoplasms, Neovascularization, Paruchuri Sailaja, Pathologic/*chemically induced/drug therapy, Phthalic Acids/pharmacology, Proceedings of the National Academy of Sciences of the United States of America, Receptors, Teegala Lakshminarayan Reddy, Thodeti Charles K
Understanding Bile Acid Signaling in Diabetes: From Pathophysiology to Therapeutic Targets
Tags: 2019, Bile Acids and Salts, Chiang John Y L, Cytoplasmic and Nuclear, Department of Integrative Medical Sciences, Diabetes & Metabolism Journal, Ferrell Jessica M, G-protein-coupled, Gastrointestinal Microbiome, June 2019 Update, NEOMED College of Medicine, Non-alcoholic Fatty Liver Disease, Receptors
Understanding Bile Acid Signaling in Diabetes: From Pathophysiology to Therapeutic Targets.
Tags: 2019, BILE acids, Bile Acids and Salts, Chiang John Y L, cholesterol 7-alpha-hydroxylase, Cytoplasmic and Nuclear, Department of Integrative Medical Sciences, Diabetes & Metabolism Journal, Endocrinology & Metabolism, Farnesoid X receptor, farnesoid-x-receptor, Fatty Liver, fatty liver-disease, Ferrell Jessica M, G protein coupled receptors, G-protein-coupled, Gastrointestinal Microbiome, growth-factor 19, gut microbiota, hepatic steatosis, improves insulin sensitivity, Liver disease, Metabolic, NEOMED College of Medicine, Non-alcoholic fatty, Non-alcoholic Fatty Liver Disease, nuclear, Receptor, Receptors, September 2019 Update, serum fgf21 levels, Syndrome
Transgenic Expression of Osteoactivin/gpnmb Enhances Bone Formation In Vivo and Osteoprogenitor Differentiation Ex Vivo.
Tags: 2016, Abdelmagid Samir M, Animals, Barbe Mary F, Bone and Bones/*metabolism, Bone Density/physiology, Bone Remodeling/genetics/*physiology, Bone Resorption/metabolism, Cell Differentiation/genetics/*physiology, Department of Anatomy & Neurobiology, Eye Proteins/genetics/*metabolism, Frara Nagat, Journal of cellular physiology, Membrane Glycoproteins/genetics/*metabolism, Mice, Moussa Fouad M, NEOMED College of Medicine, Osteoblasts/*cytology, Osteoclasts/*cytology, Osteogenesis/genetics, Owen Thomas A, Popoff Steven N, Protein-Serine-Threonine Kinases/metabolism, Receptor, Receptors, Safadi Fayez F, Sondag Gregory R, Transforming Growth Factor beta/metabolism, Transforming Growth Factor-beta Type I, Transgenic, Yingling Vanessa R
Aldo-keto reductase 1B7 is a target gene of FXR and regulates lipid and glucose homeostasis.
Tags: *Aldehyde Reductase/genetics/metabolism, 2011, Adenoviridae, Animal, Animals, Blood Glucose/*metabolism, Chiang John Y L, Cholesterol/analysis, Cytoplasmic and Nuclear/genetics/*metabolism, Department of Integrative Medical Sciences, Diabetes Mellitus/genetics/*metabolism/physiopathology, Disease Models, Fatty Liver/genetics/*metabolism/physiopathology, Ge Xuemei, Gene Expression, Genetic Vectors, Gluconeogenesis/genetics, Homeostasis, Humans, Journal of lipid research, Li Tiangang, Liver/*metabolism/physiopathology, Ma Huiyan, Malondialdehyde/blood, Mice, NEOMED College of Medicine, Polymerase Chain Reaction, Receptors, Transfection, Transgenic, Triglycerides/analysis, Yin Liya, Zhang Yanqiao
Rationally designed multi-targeted agents against neurodegenerative diseases.
Tags: 2013, Amyloid beta-Peptides/antagonists & inhibitors, Animals, Calcium Channel Blockers/chemistry/pharmacology, Cholinesterase Inhibitors/chemistry/pharmacology, Current medicinal chemistry, Drug Discovery/*methods, Geldenhuys W J, Humans, Molecular Targeted Therapy/methods, Monoamine Oxidase Inhibitors/chemistry/pharmacology, N-Methyl-D-Aspartate/antagonists & inhibitors, Neurodegenerative Diseases/*drug therapy/metabolism, Receptors, Signal Transduction/drug effects, Van der Schyf C J
Exploring Adenosine Receptor Ligands: Potential Role in the Treatment of Cardiovascular Diseases.
Tags: *drug discovery, *Ligands, 2017, Adenosine/metabolism, Animals, Atherosclerosis, Cardiac death, Cardiovascular Diseases/drug therapy/metabolism, Cardiovascular System/metabolism, Department of Integrative Medical Sciences, Geldenhuys Werner J, Hanif Ahmad, Humans, Hydrogen Bonding, Models, Molecular, Molecular Structure, Molecules (Basel, Switzerland), myocardial infarction, Nayeem Mohammed A, NEOMED College of Medicine, Protein Binding, Purinergic P1/*chemistry/*metabolism, Receptors, Signal Transduction, Structure-Activity Relationship, Vascular tone, Yun June
Virtual screening to identify novel antagonists for the G protein-coupled NK3 receptor.
Tags: *Models, *Narcotic Antagonists, *Quantitative Structure-Activity Relationship, 2010, Animals, Binding, Calcium Signaling/drug effects, CHO Cells, Competitive, Cricetinae, Cricetulus, Databases, Factual, Geldenhuys Werner J, Humans, Journal of medicinal chemistry, Kuzenko Stephanie R, Ligands, Molecular, Neurokinin-3/*antagonists & inhibitors/chemistry, Opioid/chemistry, Quinolines/*chemistry/pharmacology, Radioligand Assay, Receptors, Simmons Mark A
Structure-activity relationships of pentacycloundecylamines at the
Tags: 2007, Amines/chemical synthesis/chemistry/*pharmacology, Animals, Bioorganic & medicinal chemistry, Bloomquist Jeffrey R, Brain/drug effects, Dizocilpine Maleate/pharmacology, Excitatory Amino Acid Antagonists/*pharmacology, Geldenhuys Werner J, Inbred ICR, Ion Channels, Malan Sarel F, Male, Mice, Models, Molecular, N-Methyl-D-Aspartate/*antagonists & inhibitors, Phencyclidine/analogs & derivatives, Piperidines/pharmacology, Radioligand Assay, Receptors, Structure-Activity Relationship, Synaptosomes/*drug effects, Thiophenes/pharmacology, Van der Schyf Cornelis J
3D-QSAR and docking studies on transforming growth factor (TGF)-beta receptor 1 antagonists.
3D-QSAR and docking studies of pentacycloundecylamines at the sigma-1 (sigma1) receptor.
Tags: *Quantitative Structure-Activity Relationship, 2013, Amines/*chemistry/metabolism, Aza Compounds/chemistry, Binding Sites, Bioorganic & medicinal chemistry letters, Geldenhuys Werner J, Kinetics, Malan Sarel F, Molecular Docking Simulation, Novotny Nicholas, Protein Binding, Protein Structure, Receptors, sigma/*chemistry/metabolism, Tertiary, Van der Schyf Cornelis J
3D-Quantitative structure-activity relationship and docking studies of the tachykinin NK3 receptor.
Tags: *Quantitative Structure-Activity Relationship, 2011, Binding Sites, Bioorganic & medicinal chemistry letters, Computer Simulation, Drug Design, Geldenhuys Werner J, Humans, Ligands, Models, Molecular, Neurokinin-3/*chemistry/metabolism, Protein Structure, Quinolines/chemistry, Receptors, Simmons Mark A, Tertiary
The serotonin 5-HT6 receptor: a viable drug target for treating cognitive deficits in Alzheimer's disease.
Tags: 2009, Alzheimer Disease/*complications, Animals, Biological, Cognition Disorders/*drug therapy/*etiology, Drug Design, Expert review of neurotherapeutics, Geldenhuys Werner J, Humans, Models, Receptors, Serotonin Antagonists/chemistry/*therapeutic use, Serotonin/*metabolism, Structure-Activity Relationship, Van der Schyf Cornelis J
Role of serotonin in Alzheimer's disease: a new therapeutic target?
Tags: 2011, Alzheimer Disease/*drug therapy/*metabolism, Alzheimer's Disease – Drug Therapy, Alzheimer's Disease – Metabolism, Animals, Cell Surface – Metabolism, Clinical Trials, Clinical Trials as Topic, CNS drugs, Drug Evaluation, Geldenhuys Werner J, Humans, Preclinical, Receptors, Serotonin – Pharmacodynamics, Serotonin – Therapeutic Use, Serotonin/*metabolism, Serotonin/*pharmacology/*therapeutic use, Van der Schyf Cornelis J
Serotonin 5-HT6 receptor antagonists for the treatment of Alzheimer's disease.
Glutamate and metabotropic glutamate receptors associated with innervation of the uterine cervix during pregnancy: receptor antagonism inhibits c-Fos expression in rat lumbosacral spinal cord at parturition.
Tags: 2007, Animals, Cervix Uteri/*innervation, Department of Anatomy & Neurobiology, Excitatory Amino Acid Antagonists/pharmacology, Female, Ganglia, Gene Expression Regulation/drug effects/*physiology, Ghosh Chaitali, Glutamates/*metabolism, Hafemeister Jen, Journal of neuroscience research, Lumbosacral Region, Messenger/biosynthesis, Metabotropic Glutamate 5, Metabotropic Glutamate/*metabolism, Miller Kenneth E, NEOMED College of Medicine, Neurons/drug effects, Oncogene Proteins v-fos/metabolism, Papka Raymond E, Parturition/*metabolism, Pregnancy/*metabolism, Pyridines/pharmacology, Rats, Receptor, Receptors, Reverse Transcriptase Polymerase Chain Reaction/methods, RNA, Spinal Cord/drug effects/*physiology, Spinal/cytology, Sprague-Dawley, Storey-Workley Megan, Usip Sharon, Vesicular Glutamate Transport Protein 1/metabolism
Role of HCO3- ions in depolarizing GABAA receptor-mediated responses in pyramidal cells of rat hippocampus.
Tags: 1993, Afferent Pathways/physiology, Animals, Bicarbonates/*metabolism, Culture Techniques, Electric Stimulation, GABA-A/*physiology, gamma-Aminobutyric Acid/physiology, Grover L M, Hippocampus/*physiology, Interneurons/physiology, Journal of neurophysiology, Lambert N A, Membrane Potentials/physiology, Neurons/physiology, Rats, Receptors, Schwartzkroin P A, Synapses/physiology, Synaptic Transmission/*physiology, Teyler T J
Presynaptic mechanism for heterosynaptic, posttetanic depression in area CA1 of rat hippocampus.
Tags: 1993, Afferent/drug effects, Animals, Electric Stimulation, Electrophysiology, Evoked Potentials/physiology, Glutamate/drug effects, Glutamates/pharmacology, Glutamic Acid, Grover L M, Hippocampus/drug effects/*physiology, In Vitro Techniques, Membrane Potentials/physiology, N-Methyl-D-Aspartate/antagonists & inhibitors, Neuronal Plasticity/drug effects/physiology, Neurons, Presynaptic/drug effects/*physiology, Pyramidal Cells/drug effects, Rats, Receptors, Synapse (New York, N.Y.), Synapses/drug effects/*physiology, Teyler T J
N-methyl-D-aspartate receptor-independent long-term potentiation in area CA1 of rat hippocampus: input-specific induction and preclusion in a non-tetanized pathway.
Tags: 1992, 2-Amino-5-phosphonovalerate/*pharmacology, Animals, Electron, Evoked Potentials/drug effects, Grover L M, Hippocampus/*physiology, In Vitro Techniques, Microscopy, N-Methyl-D-Aspartate/*physiology, N-Methylaspartate/*pharmacology, Neuroscience, Pyramidal Tracts/drug effects/*physiology, Rats, Receptors, Teyler T J, Time Factors
Two components of long-term potentiation induced by different patterns of afferent activation.
Tags: 1990, 2-Amino-5-phosphonovalerate/*pharmacology, Afferent Pathways/physiology, Animals, Calcium/*physiology, Grover L M, Hippocampus/*physiology, In Vitro Techniques, Membrane Potentials, Memory/*physiology, N-Methyl-D-Aspartate/*physiology, Nature, Neuronal Plasticity, Receptors, Synaptic Transmission, Teyler T J, Time Factors
Differential effects of NMDA receptor antagonist APV on tetanic stimulation induced and calcium induced potentiation.
Tags: 1990, 2-Amino-5-phosphonovalerate/*pharmacology, Action Potentials/drug effects, Animals, Calcium/*pharmacology, Electric Stimulation, Grover L M, Hippocampus/drug effects/*physiology, In Vitro Techniques, N-Methyl-D-Aspartate, Neuronal Plasticity/*drug effects, Neuroscience letters, Neurotransmitter/antagonists & inhibitors/*physiology, Receptors, Teyler T J
Intrinsic plasticity induced by group II metabotropic glutamate receptors via enhancement of high-threshold KV currents in sound localizing neurons.
Tags: 2016, Acoustic Stimulation/methods, Action Potentials/drug effects/physiology, Animals, Auditory Pathways/drug effects/*physiology, Brain/drug effects/physiology, Chick Embryo, Department of Anatomy & Neurobiology, Glutamic Acid/metabolism, Hamlet W R, Lu Y, metabotropic glutamate receptor, Metabotropic Glutamate/agonists/*metabolism, NEOMED College of Medicine, neuromodulation, Neuronal Plasticity/drug effects/*physiology, Neurons/drug effects/*physiology, Neuroscience, nucleus laminaris, Patch-Clamp Techniques, Potassium Channels, Potassium/metabolism, Protein Kinase C/metabolism, Receptors, Sound Localization/drug effects/*physiology, Tissue Culture Techniques, Type C Phospholipases/metabolism, voltage-gated potassium channel, Voltage-Gated/*metabolism
Mechanism of vitamin D receptor inhibition of cholesterol 7alpha-hydroxylase gene transcription in human hepatocytes.
Tags: 2009, Base Sequence, Calcitriol/drug effects/genetics/*physiology, Cell Line, Cells, Chiang John Y L, Cholesterol 7-alpha-Hydroxylase/*genetics, Cultured, Department of Integrative Medical Sciences, DNA Primers, Drug metabolism and disposition: the biological fate of chemicals, Electrophoretic Mobility Shift Assay, Gene Knockdown Techniques, Genetic/*physiology, Han Shuxin, Hepatocytes/*drug effects/enzymology, Humans, Immunoprecipitation, Lithocholic Acid/pharmacology, Messenger/genetics, NEOMED College of Medicine, Polymerase Chain Reaction, Receptors, RNA, Small Interfering, Transcription, Tumor, Two-Hybrid System Techniques
A novel bile acid-activated vitamin D receptor signaling in human hepatocytes.
Tags: 2010, Calcitriol/*metabolism, Calcitriol/pharmacology, Cell Membrane/drug effects/metabolism, Cell Nucleus/drug effects/metabolism, Chiang John Y L, Cholesterol 7-alpha-Hydroxylase/antagonists & inhibitors/genetics, Department of Integrative Medical Sciences, Ellis Ewa, Enzyme Activation/drug effects, Extracellular Signal-Regulated MAP Kinases/antagonists & inhibitors, Genetic/genetics, Han Shuxin, Hep G2 Cells, Hepatocyte Nuclear Factor 4/metabolism, Hepatocytes/*drug effects/enzymology/*metabolism, Humans, Intracellular Space/drug effects/metabolism, Li Tiangang, Ligands, Lithocholic Acid/*pharmacology, Mitogen-Activated Protein Kinase Kinases/metabolism, Molecular endocrinology (Baltimore, Md.), NEOMED College of Medicine, Phosphorylation/drug effects, Phosphotyrosine/metabolism, Promoter Regions, Protein Kinase Inhibitors/pharmacology, Protein Transport/drug effects, Proto-Oncogene Proteins c-raf/metabolism, Receptors, Retinoid X Receptor alpha/metabolism, Signal Transduction/*drug effects, src-Family Kinases/metabolism, Steroid Hydroxylases/genetics/metabolism, Strom Stephen, Vitamin D3 24-Hydroxylase
Reduced AMPK activation and increased HCAR activation drive anti-inflammatory response and neuroprotection in glaucoma.
Tags: 2018, AMP-activated protein kinase, AMP-Activated Protein Kinases/*metabolism, Animal, Animals, Biological, Calcium Binding Proteins – Metabolism, Calcium-Binding Proteins/metabolism, Cells – Drug Effects, Cells – Pathology, Department of Pharmaceutical Sciences, Diet, Disease Models, Eye Proteins/genetics, Female, G-Protein-Coupled – Metabolism, G-Protein-Coupled/*metabolism, Glaucoma, Glaucoma – Complications, Glaucoma – Pathology, Glaucoma/*complications/pathology, Harun-Or-Rashid Mohammad, Impact of Events Scale, Inbred DBA, Inflammation – Etiology, Inflammation – Prevention and Control, Inflammation hydroxycarboxylic acid receptor, Inflammation/*etiology/*prevention & control, Inman Denise M, Journal of neuroinflammation, Ketogenic diet, Ketogenic/methods, Male, Membrane Glycoproteins, Membrane Glycoproteins/genetics, Mice, Microfilament Proteins – Metabolism, Microfilament Proteins/metabolism, Microglia/drug effects/pathology, Models, Mutation, Mutation/genetics, NEOMED College of Pharmacy, Neuroprotection/drug effects/*physiology, NLR Family, Optic Nerve – Pathology, Optic Nerve/pathology, Phosphotransferases – Metabolism, Proteins, Pyrin Domain-Containing 3 Protein/genetics/metabolism, Receptors, Retina – Drug Effects, Retina – Pathology, Retinal Ganglion Cells/drug effects/*pathology, Transgenic
Integrin mediated adhesion of osteoblasts to connective tissue growth factor (CTGF/CCN2) induces cytoskeleton reorganization and cell differentiation.
Tags: *Cell Differentiation, 2015, Animals, Barbe Mary F, Cell Adhesion, Cell Line, Connective Tissue Growth Factor/chemistry/*metabolism, Core Binding Factor Alpha 1 Subunit/metabolism, Cytoskeleton/*metabolism, Department of Anatomy & Neurobiology, Extracellular Signal-Regulated MAP Kinases/metabolism, Focal Adhesion Protein-Tyrosine Kinases/metabolism, Hendesi Honey, Integrins/*metabolism, Mice, Monroy M Alexandra, NEOMED College of Medicine, Osteoblasts/*cytology/*metabolism, PloS one, Popoff Steven N, rac GTP-Binding Proteins/metabolism, Receptors, Safadi Fayez F, Signal Transduction, Transcriptional Activation, Vitronectin/metabolism
The effects of aging on mu and delta opioid receptors in the spinal cord of Fischer-344 rats.
Tags: 1998, Aging/*metabolism, Ala(2)-MePhe(4)-Gly(5)-, Animals, Brain research, Crisp T, delta/antagonists & inhibitors/*metabolism, Enkephalin, Enkephalins/metabolism, Gordon T L, Hoskins D L, Inbred F344, Male, mu/agonists/*metabolism, Naltrexone/analogs & derivatives/metabolism, Narcotic Antagonists/metabolism, Opioid, Radioligand Assay, Rats, Receptors, Spinal Cord/*metabolism
Reduced vascular responsiveness after a single bout of dynamic exercise in the conscious rabbit.
Tags: 1992, Adenosine/pharmacology, Adrenergic/physiology, Animals, Blood Vessels/*physiology, DiCarlo S E, Dose-Response Relationship, Drug, Hindlimb/physiology, Howard M G, In Vitro Techniques, Isoproterenol/pharmacology, Journal of applied physiology (Bethesda, Md. : 1985), Phenylephrine/pharmacology, Physical Exertion/*physiology, Pressoreceptors/physiology, Purinergic/physiology, Rabbits, Receptors, Reflex/physiology, Regional Blood Flow/physiology